TM30089(TM 30089)|CRTH2 antagonist|DC Chemicals

Cas No.:	844639-57-2
Chemical Name:	2-[3-[(4-fluorophenyl)sulfonyl-methylamino]-1,2,3,4-tetrahydrocarbazol-9-yl]aceticacid
Synonyms:	TM 30089,TM-30089
SMILES:	O=C(O)CN1C2=C(C3=C1C=CC=C3)CC(N(S(=O)(C4=CC=C(F)C=C4)=O)C)CC2
Formula:	C₂₁H₂₀FN₂O₄S∙Na
M.Wt:	438.45
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

TM30089 is a slective CRTH2 antagonist, displaying high antagonistic potency on mouse CRTH2 with low affinity to TP and many other prostanoid receptors including the related anaphylatoxin C3a and C5a receptors.For the detailed information of TM30089, the solubility of TM30089 in water, the solubility of TM30089 in DMSO, the solubility of TM30089 in PBS buffer, the animal experiment (test) of TM30089, the cell expriment (test) of TM30089, the in vivo, in vitro and clinical trial test of TM30089, the EC50, IC50,and Affinity of TM30089, Please contact DC Chemicals.

MSDS

COA

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2018-0101

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