Α5ia (α5IA)|cas 215874-86-5|buy|Price|from DC Chemicals

Cas No.:	215874-86-5
Chemical Name:	1,2,4-Triazolo[3,4-a]phthalazine, 3-(5-methyl-3-isoxazolyl)-6-[(1-methyl-1H-1,2,3-triazol-4-yl)methoxy]-
Synonyms:	Α5ia
SMILES:	CC1=CC(=NO1)C2=NN=C3N2N=C(C4=CC=CC=C43)OCC5=CN(N=N5)C
Formula:	C₁₇H₁₄N₈O₂
M.Wt:	362.35
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

α5IA is a selective inverse agonist For Α5 subtype of GABAA receptor with a higher intrinsic activity at the A5 subtype than other drugs. α5IA enhances cognition in laboratory animals without being proconvulsant or anxiogenic. α5IA acts as an "alcohol antagonist," markedly reducing the amnesic effect of alcohol and partially attenuating sedation, similar to Ro15-4513, but without the anxiogenic effect. α5IA offers promise as a tool to study cognitive disorders, memory function, and treatment of alcohol-related disorders.For the detailed information of Α5ia (α5IA), the solubility of Α5ia (α5IA) in water, the solubility of Α5ia (α5IA) in DMSO, the solubility of Α5ia (α5IA) in PBS buffer, the animal experiment (test) of Α5ia (α5IA), the cell expriment (test) of Α5ia (α5IA), the in vivo, in vitro and clinical trial test of Α5ia (α5IA), the EC50, IC50,and Affinity of Α5ia (α5IA), Please contact DC Chemicals.

MSDS

COA

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2018-0101

Cat. No.	Product name	Field of application
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