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TP-1454

  Cat. No.:  DC72893   Featured
Chemical Structure
2490276-04-3
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More than 5000 active chemicals with high quality for research!
Field of application
TP-1454 is an activator of PKM2 with AC50 of 10 Nm in biochemical assays.TP-1454 modulates tumor-immune responses by destabilizing T-regulatory cells.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2490276-04-3
Chemical Name: 1H-Pyrazole-5-carboxamide, N-[(2-amino-6-fluorophenyl)methyl]-N-[2-(tetrahydro-1,1-dioxido-2H-thiopyran-4-yl)ethyl]-3-(trifluoromethyl)-
Synonyms: 1H-Pyrazole-5-carboxamide, N-[(2-amino-6-fluorophenyl)methyl]-N-[2-(tetrahydro-1,1-dioxido-2H-thiopyran-4-yl)ethyl]-3-(trifluoromethyl)-
SMILES: N1C(C(N(CC2=C(F)C=CC=C2N)CCC2CCS(=O)(=O)CC2)=O)=CC(C(F)(F)F)=N1
Formula: C19H22F4N4O3S
M.Wt: 462.46
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: TP-1454 is an activator of PKM2 with AC50 of 10 Nm in biochemical assays.TP-1454 modulates tumor-immune responses by destabilizing T-regulatory cells.
MSDS
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