DCC3474 |
Mrgx1-activator-1 |
Activator of MrgX1 receptor signaling |
|
DCC3475 |
Mri-1891 |
Novel peripheral CB1R antagonist, being highly biased toward inhibiting CB1R-induced β-arrestin-2 (βArr2) recruitment over G-protein activation |
|
DCC3476 |
Mrl-248 |
Novel potent and selective RORγT inhibitor, showing no appreciable activity against a panel of related nuclear hormone receptors |
|
DCC3477 |
Mrl-299 |
Novel potent RORγT inhibitor |
|
DCC3478 |
Mrl-367 |
Novel potent and selective RORγT inhibitor, showing no appreciable activity against a panel of related nuclear hormone receptors |
|
DCC3479 |
Mrl-770 |
Novel selective and reproducible inhibitor of DNA synthesis in E. coli JL553 |
|
DCC3480 |
Mrs2220 |
Selective enhancer of the ATP effects at fast desensitizing P2X (P2X1 and P2X3) receptors |
|
DCC3481 |
mrs2690 |
Potent P2Y14 receptor agonist |
|
DCC3482 |
mrs2693 Trisodium |
Selective P2Y6 agonist |
|
DCC3483 |
mrs2768 |
Selective P2Y2 agonist |
|
DCC3484 |
mrs2957 |
Potent P2Y6 agonist |
|
DCC3485 |
Mrs2964 |
Potent and selective P2Y6 receptor agonist |
|
DCC3486 |
Mrs4598 |
Novel highly potent human CD73 inhibitor (K i = 0.673 nM) |
|
DCC3487 |
Mrs4608 |
Novel potent antagonist of P2Y 14 receptor (P2Y 14 R) (IC 50 ~20 nM at hP2Y 14 R/mP2Y 14 R) |
|
DCC3488 |
Mrs4654 |
Novel potent P2Y14 Receptor Antagonist (IC 50 , 15 nM) |
|
DCC3489 |
Mrs7396 |
Bitopic fluorescent antagonist of the A2A adenosine receptor |
|
DCC3490 |
Mrs7469 |
Novel highly selective A1 adenosine receptor (A1AR) agonist |
|
DCC3491 |
Mrs7591 |
Novel Partial Agonist of Human and Mouse A3 Adenosine Receptors (Ki = 10.9/17.8 nM, at human/mouse A3AR) |
|
DCC3492 |
Mrs7799 |
Novel highly potent A3 adenosine receptor (A3AR) antagonist with Kd values (nM): 0.55 (human), 3.74 (mouse), and 2.80 (rat) |
|
DCC3493 |
Mrt-68601 Hydrochloride |
Potent inhibitor of TANK-binding kinase-1 (TBK1)/IKKepislon kinases |
|
DCC3494 |
Mrt-92 Hydrochloride |
Novel inhibitor of Hedgehog signaling by blocking overlapping binding sites in the transmembrane domain of the Smoothened receptor |
|
DCC3495 |
Mrz-8676 |
Novel, selective, orally bioavailable, negative allosteric modulator of subtype 5 metabotropic glutamate receptors (mGluR5) |
|
DCC3496 |
ms0017509 |
Inhibitor of DNA damage repair |
|
DCC3497 |
ms0019266 |
Novel inhibitor of DNA damage repair |
|
DCC3498 |
Ms2126 |
Novel inhibitor of Human p53 and CREB Binding Protein (CREBBP) interaction |
|
DCC3499 |
Ms2177 |
Novel potent and selective SETD8 inhibitor |
|
DCC3500 |
Ms2i6a |
Mitochondrial tRNA-specific modification, regulating efficient mitochondrial translation and energy metabolism in mammals |
|
DCC3501 |
Msc2524070 |
Novel potent tankyrase (TNKS) inhibitor (EC 50 : 2 nM) |
|
DCC3502 |
Msc-4381 |
Novel inhibitor of SLC16A3 |
|
DCC3503 |
Msd-496486311 |
Novel potent and selective PI3Kδ inhibitor |
|