6-Benzoylheteratisine

  Cat. No.:  DC45361  
Chemical Structure
99759-48-5
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More than 5000 active chemicals with high quality for research!
Field of application
6-Benzoylheteratisine is a naturally occurring antagonist of the Na+ channel activator aconitine.
Cas No.: 99759-48-5
Chemical Name: 6-Benzoylheteratisine
SMILES: CO[C@@H]1[C@]23[C@]4([H])[C@@H]([C@@]([C@@]5([C@]6([H])[C@@]3([H])C[C@H](CC5)OC6=O)O)([H])[C@@]2([H])N(C[C@@]4(CC1)C)CC)OC(C7=CC=CC=C7)=O
Formula: C29H37NO6
M.Wt: 495.61
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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MSDS_29084_DC45361_99759-48-5
COA
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Cat. No. Product name Field of application
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DC46036 GX-201 GX-201 is a selective NaV1.7 inhibitor, with an IC50 of <3.2 nM for hNaV1.7.
DC45807 Nav1.7-IN-8 Nav1.7-IN-8 is a potent blockage of NaV1.7 with high selectivity for the inhibition of NaV1.7 over the subtypes hNaV1.1 and hNaV1.5. Nav1.7-IN-8 inhibits CYP2C9 and CYP3A4 with an IC50 of 0.17 μM and 0.077 μM, respectively. Nav1.7-IN-8 displays significant analgesic effects in rodent models of acute and inflammatory pain.
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DC45361 6-Benzoylheteratisine 6-Benzoylheteratisine is a naturally occurring antagonist of the Na+ channel activator aconitine.
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