| DC47323 |
TRPA1 Antagonist 3
|
TRPA1 Antagonist 3 is a photoswitchable TRPA1 agonist that enables optical control of the TRPA1 channel. |
| DC47322 |
4-(Phenyldiazenyl)benzoic acid
|
4-(Phenyldiazenyl)benzoic acid is a photosensitive and photoswitchable TRPA1 agonist that can be used as pharmacological tools for study of pain signaling. |
| DC47246 |
SB 452533
|
SB 452533 is a potent and selective TRPV1 antagonist with the pKb of 7.8. |
| DC46699 |
9-Phenanthrol
|
9-Phenanthrol (9-Hydroxyphenanthrene, Phenanthren-9-o, 9-Phenanthrenol) is a selective TRPM4 inhibitor with an IC50 in the range of 0.02 μM, without effects on TRPM5. |
| DC46466 |
Dihydrocapsiate
|
Dihydrocapsiate, as a compound of capsinoid family, is an orally active TRPV1 agonist. Dihydrocapsiate can be used for the research of metabolism disease. |
| DC46465 |
Capsiate
|
Capsiate, as a capsaicin analogue extracted from a non-pungent cultivar of CH-19 sweet red pepper, is an orally active agonist of TRPV1. |
| DC45871 |
Methyl kakuol
|
Methyl kakuol shows agonistic activity against TRPA1 with an EC50 of 0.27 µM. |
| DC45849 |
GSK2332255B
|
GSK2332255B is a potent, selective TRPC3 and TRPC6 antagonist with IC50s of 5 nM and 4 nM for rat TRPC3 and rat TRPC6. GSK2332255B shows ≥100-fold selectivity for TRPC3/6 over other calcium-permeable channels. |
| DC45289 |
OptoBI-1
|
OptoBI-1 is a photochromic TRPC3 agonist, which asts as a photopharmacological tool to control of neuronal firing. |
| DC45288 |
AMG2850
|
AMG2850 is a potent, orally bioavailable and selective transient receptor potential melastatin 8 (TRPM8) antagonist. |
