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TAK-615

  Cat. No.:  DC10923   Featured
Chemical Structure
1664335-55-0
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More than 5000 active chemicals with high quality for research!
Field of application
TAK-615 (TAK615) is a potent, selective, negative allosteric modulator (NAM) of the LPA1 receptor, partially inhibits the LPA response with IC50 of 91 nM (60% at 10 uM) in calcium mobilisation assays..
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1664335-55-0
Chemical Name: 4-((N-(cyclopropylmethyl)-4-(2-fluorophenoxy)benzamido)methyl)benzoic acid
Synonyms: TAK615; TAK 615
SMILES: C(O)(=O)C1=CC=C(CN(CC2CC2)C(=O)C2=CC=C(OC3=CC=CC=C3F)C=C2)C=C1
Formula: C25H22FNO4
M.Wt: 419.452
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: 1. Ellery J, et al. Eur J Pharmacol. 2018 May 26;833:8-15.
Description: TAK-615 (TAK615) is a potent, selective, negative allosteric modulator (NAM) of the LPA1 receptor, partially inhibits the LPA response with IC50 of 91 nM (60% at 10 uM) in calcium mobilisation assays.
References: References 1. Ellery J, et al. Eur J Pharmacol. 2018 May 26;833:8-15. View Related Products by Target Lysophospholipid Receptor
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
Cat. No. Product name Field of application
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DC10923 TAK-615 TAK-615 (TAK615) is a potent, selective, negative allosteric modulator (NAM) of the LPA1 receptor, partially inhibits the LPA response with IC50 of 91 nM (60% at 10 uM) in calcium mobilisation assays..
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