Elsulfavirine

  Cat. No.:  DC11892   Featured
Chemical Structure
868046-19-9
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More than 5000 active chemicals with high quality for research!
Field of application
A new-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) for the treatment of HIV-1 infections, the prodrug of the active compound VM-1500A..
Cas No.: 868046-19-9
Chemical Name: N-(4-{2-[4-bromo-3-(3-chloro-5-cyanophenoxy)- 2-fluorophenyl]acetamido}- 3-chlorobenzenesulfonyl)propanamide
Synonyms: Elpida
SMILES: C(NS(C1=CC=C(NC(=O)CC2=CC=C(Br)C(OC3=CC(C#N)=CC(Cl)=C3)=C2F)C(Cl)=C1)(=O)=O)(=O)CC
Formula: C24H17BrCl2FN3O5S
M.Wt: 626.94
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Elsulfavirine is a reverse transcriptase inhibitors for HIV-1 infection and is a new anti-HIV drug[1].
Target: HIV-1
References: [1]. Rai MA, et al. Emerging reverse transcriptase inhibitors for HIV-1 infection. Expert Opin Emerg Drugs. 2018 Jun;23(2):149-157.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
Cat. No. Product name Field of application
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DC10355 Nelfinavir Nelfinavir(AG-1341) is a potent and orally bioavailable human immunodeficiency virus HIV-1 protease inhibitor (Ki=2 nM) and is widely prescribed in combination with HIV reverse transcriptase inhibitors for the treatment of HIV infection.
DC9476 NBD-556 NBD-556 is small molecule mimetic of CD4, NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.
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