GSK256073

  Cat. No.:  DC42499  
Chemical Structure
862892-90-8
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More than 5000 active chemicals with high quality for research!
Field of application
GSK256073 is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM)and dyslipidemia. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2
Cas No.: 862892-90-8
Synonyms: GSK256073
SMILES: O=C(N(C1=C2NC(Cl)=N1)CCCCC)NC2=O
Formula: C10H13ClN4O2
M.Wt: 256.69
Sotrage: Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month
MSDS
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MSDS_26127_DC42499_862892-90-8
COA
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Cat. No. Product name Field of application
DC42499 GSK256073 GSK256073 is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM)and dyslipidemia. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2
DC9455 MK-6892 MK-6892 is a highly potential GPR109A agonist with Ki value of 4.0 nM.
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