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hA2A/hCA XII modulator 1

  Cat. No.:  DC71212  
Chemical Structure
2548963-55-7
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Field of application
hA2A/hCA XII modulator 1 (compound 14), a triazolopirazine, is a potent hA2A adenosine receptor (hA2AAR) antagonist with Kis of 6.4 nM, 4.819 μM, >30 μM for hA2AAR, hA1AR, hA3AR, respectively. hA2A/hCA XII modulator 1 is a potent human carbonic anhydrase XII (hCA XII) inhibitor with Kis of 6.2 nM, 46 nM, 466 nM, 8.351 μM for hCA XII, hCA II, hCA IX and hCA I, respectively. hA2A/hCA XII modulator 1 has the potential for cancer research.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2548963-55-7
Chemical Name: hA2A/hCA XII modulator 1
M.Wt: 501.52
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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MSDS_35438_DC71212_2548963-55-7
COA
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Cat. No. Product name Field of application
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