Paltusotine

  Cat. No.:  DC46145   Featured
Chemical Structure
2172870-89-0
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More than 5000 active chemicals with high quality for research!
Field of application
Paltusotine (CRN00808) is an orally active, nonpeptide selective somatostatin type 2 (SST2) receptor agonist. Paltusotine has the potential for maintaining GH and IGF-1 levels after depot somatostatin receptor ligand therapy.
Cas No.: 2172870-89-0
Chemical Name: Paltusotine
Synonyms: Paltusotine;F2IBD1GMD3;3-(4-(4-Aminopiperidin-1-yl)-3-(3,5-difluorophenyl)quinolin-6-yl)-2-hydroxybenzonitrile;3-[4-(4-aminopiperidin-1-yl)-3-(3,5-difluorophenyl)quinolin-6-yl]-2-hydroxybenzonitrile;Paltusotine [INN];BDBM405588;US10351547, Compound 2-2;Benzonitrile, 3-(4-(4-amino-1-piperidinyl)-3-(3,5-difluorophenyl)-6-quinolinyl)-2-hydroxy-
SMILES: FC1C([H])=C(C([H])=C(C=1[H])C1=C([H])N=C2C([H])=C([H])C(C3=C([H])C([H])=C([H])C(C#N)=C3O[H])=C([H])C2=C1N1C([H])([H])C([H])([H])C([H])(C([H])([H])C1([H])[H])N([H])[H])F
Formula: C27H22F2N4O
M.Wt: 456.4866
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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MSDS_29938_DC46145_2172870-89-0
COA
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Cat. No. Product name Field of application
DC46145 Paltusotine Paltusotine (CRN00808) is an orally active, nonpeptide selective somatostatin type 2 (SST2) receptor agonist. Paltusotine has the potential for maintaining GH and IGF-1 levels after depot somatostatin receptor ligand therapy.
DC28234 L-803087 L-803087 is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM, which is > 280-fold higher than other somatostatin receptors. L-803087 facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice.
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