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Tocainide

  Cat. No.:  DC48532   Featured
Chemical Structure
41708-72-9
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More than 5000 active chemicals with high quality for research!
Field of application
Tocainide hydrochloride is an orally activesodium channel blocker, it blocks the sodium channels in the pain-producing foci in the nerve membranes. Tocainide hydrochloride is a primary amine analog of lidocaine, can be used for the treatment of tinnitus.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 41708-72-9
Chemical Name: Tocainide
Synonyms: Tocainide;2-Amino-N-(2,6-dimethylphenyl)propanamide;N-(2-Aminopropionyl)-2,6-xylidine;2-amino-2',6'-propionoxylidide;6'-propionoxylidide,2-amino-2;alanyl-2,6-xylidide;S-Tocainide
SMILES: CC1=C(NC(C(N)C)=O)C(C)=CC=C1
Formula: C11H16N2O
M.Wt: 192.25754
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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DC48532 Tocainide Tocainide hydrochloride is an orally activesodium channel blocker, it blocks the sodium channels in the pain-producing foci in the nerve membranes. Tocainide hydrochloride is a primary amine analog of lidocaine, can be used for the treatment of tinnitus.
DC47939 NBI-921352 NBI921352 is a Nav1.6 inhibitor with an IC50 value of 3.765 μM.
DC7287 Ralfinamide Sodium channel blocker. Suppresses tetrodotoxin (TTX)-resistant Na+ currents approximately twice as selectively as TTX-sensitive currents. Antinociceptive; displays analgesic effects in animal models of inflammatory and neuropathic pain.
DC9623 Flecainide (acetate) Flecainide(Tambocor) is a class 1C antiarrhythmic drug especially used for the management of supraventricular arrhythmia; works by blocking the Nav1.5 sodium channel in the heart, causing prolongation of the cardiac action potential.
DC11649 Jamaicin (AnCoA4) AnCoA4 (AnCoA-4, AnCoA 4) is a potent Orai1 channel inhibitor that inhibits store-operated calcium (SOC) with EC50 of 0.88 uM.
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