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WDR5 inhibitor 41

  Cat. No.:  DC70902  
Chemical Structure
2417012-26-9
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More than 5000 active chemicals with high quality for research!
Field of application
WDR5 inhibitor 41 is a potent, selective and orally bioavailable WDR5 WIN-site inhibitor with TR-FRET Ki value of <0.02 nM, inhibits cell proliferation of MV4:11 and MOLM-13 with IC50 of 13 and 27 nM, respectively.WDR5 inhibitor 41 is well tolerated in mice by both iv and po dosing and showed no clinical sign of abnormalities suggesting an enhanced safetyprofile for the series.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2417012-26-9
Chemical Name: WDR5 inhibitor 41
Formula: C29H29F3N6O
M.Wt: 534.587
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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