DC72681 |
SPC4061
|
SPC4061 an antisense nucleotide, is a potent PCSK9 inhibitor. SPC4061 targets the lock-in nucleic acid (LNA) of PCSK9 for the study of hypercholesterolemia and related diseases. |
DC72680 |
PPACK II diTFA
|
PPACK II diTFA is an irreversible and specific glandular and plasma kallikreins inhibitor. |
DC72410 |
Ac-Phe-Gly-pNA
|
Ac-Phe-Gly-pNA is the chymotrypsin specific substrate. |
DC72409 |
AAF-CMK
|
AAF-CMK is a TPPII (tripeptidylpeptidase II) inhibitor, shows anti-tumor activity and induces apoptosis. AAF-CMK can be used in leukemia research. |
DC72231 |
Cyclotheonamide A
|
Cyclotheonamide A is a serine protease inhibitor (cyclic polypeptide), which can be obtained from marine sponges of the genus Theonella. Cyclotheonamide A shows potent inhibitory activity against trypsin (Ki=0.023 µM) and streptokinase (Ki=0.035 µM) and moderate inhibitory activity against human α-thrombin (Ki=0.18 µM). Cyclotheonamide A can be used in study of antithrombotic. |
DC72230 |
UAMC-00050
|
UAMC-00050 is a potent trypsin-like serine protease inhibitor. UAMC-00050 can be used in research of dry eye syndrome and ocular inflammation. |
DC71824 |
Tilpisertib fosmecarbil
|
Tilpisertib fosmecarbil is a potent serine/threonine kinase inhibitor. Tilpisertib fosmecarbil has anti-inflammatory activity. |
DC71823 |
Bezeparsen
|
Bezeparsen is a PCSK9 synthesis inhibitor. |
DC71558 |
Chymotrypsin
|
Chymotrypsin (Chymotrypsin A) is a serine protease produced by the pancreas. Chymotrypsin cleaves protein chains at the carboxyl side of aromatic amino acids. |
DC71557 |
JO146
|
JO146 is a Chlamydia trachomatis high temperature requirement A (CtHtrA) protease inhibitor with IC50s of 21.86 and 1.15 μM for CtHtrA and human neutrophil elastase (HNE), respectively. JO146 can be used to inhibits bacterial infections. |