Cat. No. | Product name | CAS No. |
DC11270 |
MSX-130
Featured
MSX-130 is CXCR4 Antagonist. |
4051-59-6 |
DC10023 |
MT-1
Featured
MT1 is a bivalent chemical probe of BET bromodomains.MT1 is an intramolecular bivalent BRD4 binder that is more than 100-fold more potent, in cellular assays, than the corresponding monovalent antagonist, JQ1. |
|
DC22167 |
MT-802
Featured
MT-802 (MT802) is a potent BTK PROTAC that induces degradation of both wild-type and C481S mutant BTK (DC50=9.1 nM). |
2231744-29-7 |
DC10332 |
Methylthio-DADMe-Immucillin A; MTDIA
Featured
MT-DADMe-ImmA is an inhibitor of human 5'-methylthioadenosine phosphorylase (MTAP) with a Ki of 90 pM. |
653592-04-2 |
DC22139 |
MTI-31
Featured
MTI31 (LXI-15029, mTOR inhibitor-31) is a novel potent, selective mTORC1/mTORC2 inhibitor with Kd of 0.2 nM (mTOR), displays >5,000-fold selectivity over PIK3CA, PIK3CB and PIK3G. |
1567915-38-1 |
DC20230 |
mTOR inhibitor-1
Featured
mTOR inhibitor-1 is a novel mTOR pathway inhibitor which can suppress cells proliferation and inducing autophagy. |
468747-17-3 |
DC8240 |
3-(4,5-Dimethylthiazol-2-yl)-5-(3-carboxymethoxyphenyl)-2-(4-sulfophenyl)-2H-tetrazolium
Featured
MTS is water-soluble and used in the MTS assay. |
138169-43-4 |
DC10871 |
MTX211
Featured
MTX-211 is a dual inhibitor of EGFR and PI3K, used for the treatment of cancer and other diseases. |
1952236-05-3 |
DC7205 |
Mubritinib (TAK 165)
Featured
Mubritinib is a potent inhibitor of the human epidermal growth factor receptor 2 (HER2) tyrosine kinase. |
366017-09-6 |
DC11273 |
Murepavadin (POL7080)
Featured
Murepavadin is a novel class of highly specific outer membrane protein targeting antibiotic to treat resistant Pseudomonas infections. |
944252-63-5 |
DC10915 |
mutant EGFR inhibitor B30
Featured
mutant EGFR inhibitor B30 is a potent, selective, next-generation EGFR mutants inhibitor with IC50 of 1.1 and 7.2 nM for EGFRL858R and EGFRL858R/T790M/C797S, respectively. |
2225887-26-1 |
DC7982 |
Mutant IDH1-IN-1
Featured
Mutant IDH1-IN-1 is a potent mutant IDH1 R132H inhibitor with IC50 < 0.1 uM(A level in Patent). |
1355326-21-4 |
DC11829 |
MW-150
Featured
MW-150 is a novel potent, selective, CNS penetrant and orally active inhibitor of p38α MAPK with Ki of 101 nM |
1628502-91-9 |
DC26051 |
MX1013
Featured
MX1013 is a dipeptide pan-caspase inhibitor that inhibits caspase-1 |
582316-00-5 |
DC10074 |
MX69
Featured
MX69 is the MDM2/XIAP inhibitor, used for cancer treatment. |
1005264-47-0 |
DC10952 |
MYCMI-6(NSC 354961)
Featured
MYCMI-6 (NSC354961) is a selective, high affinity inhibitor of MYC-MAX interaction, blocks MYC-driven transcription and binds selectively to the MYC bHLHZip domain with Kd of 1.6 uM in SPR assay. |
681282-09-7 |
DC10606 |
Mycro-3
Featured
Mycro 3 is potent and selective for c-Myc in whole cell assays. |
944547-46-0 |
DC21360 |
MZ1
Featured
MZ1 is a PROTAC that tethers JQ1 to a ligand for the E3 ubiquitin ligase VHL, triggers, induces degradation of the BET bromodomain BRD4. |
1797406-69-9 |
DC9298 |
thiotepa
Featured
N,N’N’-triethylenethiophosphoramide (ThioTEPA) is a cancer chemotherapeutic member of the alkylating agent group. |
52-24-4 |
DC8271 |
NSC-41589
Featured
N-[2-(methylsulfanyl) phenyl]acetamide. |
6310-41-4 |
DC10159 |
N3-PEG3-vc-PAB-MMAE
Featured
N3-PEG3-vc-PAB-MMAE is a drug-linker conjugate for ADC with potent antitumor activity by using the anti-mitotic agent, monomethyl auristatin E (MMAE), linked via the peptide N3-PEG3-vc-PAB. |
|
DC7471 |
N6022
Featured
N6022 is a potent, selective, reversible, and efficacious S-Nitrosoglutathione reductase(GSNOR) inhibitor(IC50=10 nM) which is currently undergoing clinical development. |
1208315-24-5 |