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Cat. No. Product name CAS No.
DC11270 MSX-130 Featured

MSX-130 is CXCR4 Antagonist.

4051-59-6
DC10023 MT-1 Featured

MT1 is a bivalent chemical probe of BET bromodomains.MT1 is an intramolecular bivalent BRD4 binder that is more than 100-fold more potent, in cellular assays, than the corresponding monovalent antagonist, JQ1.

DC22167 MT-802 Featured

MT-802 (MT802) is a potent BTK PROTAC that induces degradation of both wild-type and C481S mutant BTK (DC50=9.1 nM).

2231744-29-7
DC10332 Methylthio-DADMe-Immucillin A; MTDIA Featured

MT-DADMe-ImmA is an inhibitor of human 5'-methylthioadenosine phosphorylase (MTAP) with a Ki of 90 pM.

653592-04-2
DC22139 MTI-31 Featured

MTI31 (LXI-15029, mTOR inhibitor-31) is a novel potent, selective mTORC1/mTORC2 inhibitor with Kd of 0.2 nM (mTOR), displays >5,000-fold selectivity over PIK3CA, PIK3CB and PIK3G.

1567915-38-1
DC20230 mTOR inhibitor-1 Featured

mTOR inhibitor-1 is a novel mTOR pathway inhibitor which can suppress cells proliferation and inducing autophagy.

468747-17-3
DC8240 3-(4,5-Dimethylthiazol-2-yl)-5-(3-carboxymethoxyphenyl)-2-(4-sulfophenyl)-2H-tetrazolium Featured

MTS is water-soluble and used in the MTS assay.

138169-43-4
DC10871 MTX211 Featured

MTX-211 is a dual inhibitor of EGFR and PI3K, used for the treatment of cancer and other diseases.

1952236-05-3
DC7205 Mubritinib (TAK 165) Featured

Mubritinib is a potent inhibitor of the human epidermal growth factor receptor 2 (HER2) tyrosine kinase.

366017-09-6
DC11273 Murepavadin (POL7080) Featured

Murepavadin is a novel class of highly specific outer membrane protein targeting antibiotic to treat resistant Pseudomonas infections.

944252-63-5
DC10915 mutant EGFR inhibitor B30 Featured

mutant EGFR inhibitor B30 is a potent, selective, next-generation EGFR mutants inhibitor with IC50 of 1.1 and 7.2 nM for EGFRL858R and EGFRL858R/T790M/C797S, respectively.

2225887-26-1
DC7982 Mutant IDH1-IN-1 Featured

Mutant IDH1-IN-1 is a potent mutant IDH1 R132H inhibitor with IC50 < 0.1 uM(A level in Patent).

1355326-21-4
DC11829 MW-150 Featured

MW-150 is a novel potent, selective, CNS penetrant and orally active inhibitor of p38α MAPK with Ki of 101 nM

1628502-91-9
DC26051 MX1013 Featured

MX1013 is a dipeptide pan-caspase inhibitor that inhibits caspase-1

582316-00-5
DC10074 MX69 Featured

MX69 is the MDM2/XIAP inhibitor, used for cancer treatment.

1005264-47-0
DC10952 MYCMI-6(NSC 354961) Featured

MYCMI-6 (NSC354961) is a selective, high affinity inhibitor of MYC-MAX interaction, blocks MYC-driven transcription and binds selectively to the MYC bHLHZip domain with Kd of 1.6 uM in SPR assay.

681282-09-7
DC10606 Mycro-3 Featured

Mycro 3 is potent and selective for c-Myc in whole cell assays.

944547-46-0
DC21360 MZ1 Featured

MZ1 is a PROTAC that tethers JQ1 to a ligand for the E3 ubiquitin ligase VHL, triggers, induces degradation of the BET bromodomain BRD4.

1797406-69-9
DC9298 thiotepa Featured

N,N’N’-triethylenethiophosphoramide (ThioTEPA) is a cancer chemotherapeutic member of the alkylating agent group.

52-24-4
DC8271 NSC-41589 Featured

N-[2-(methylsulfanyl) phenyl]acetamide.

6310-41-4
DC10159 N3-PEG3-vc-PAB-MMAE Featured

N3-PEG3-vc-PAB-MMAE is a drug-linker conjugate for ADC with potent antitumor activity by using the anti-mitotic agent, monomethyl auristatin E (MMAE), linked via the peptide N3-PEG3-vc-PAB.

DC7471 N6022 Featured

N6022 is a potent, selective, reversible, and efficacious S-Nitrosoglutathione reductase(GSNOR) inhibitor(IC50=10 nM) which is currently undergoing clinical development.

1208315-24-5
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