DCC4226 |
Ppk1-in-8 |
Novel PPK1 inhibitor, preventing UTI effectively through the disruption of the PPK1 function |
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DCC4227 |
pppone |
Potent and selective antagonist of melanocortin-4 receptor (MC4R) |
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DCC4228 |
Ppq-581 |
Novel anti-influenza agent, interrupting the crucial RNP trafficking, resulting in influenza replication inhibition, preventing virus-induced cytopathic effects |
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DCC4229 |
Ppt (water-heme Modulator) |
Novel Modulator of Water-Heme Interactions in Low-Spin P450 Complexes of CYP2C9d and CYP125A1 |
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DCC4230 |
Ppxy Budding Inhibitor 4 |
Novel inhibitor of budding of mVP40 and eVP40 VLPs, blocking mVP40-795 Nedd4 protein-protein interaction. |
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DCC4231 |
Ppxy Budding Inhibitor 5 |
Specific blocker of the MARV VP40 PPxY-host Nedd4 interaction and subsequent PPxY-dependent egress of MARV VP40 VLPs. |
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DCC4232 |
Pqa-11 |
Novel potent neuroprotectant, inhibiting glutamate-induced cell death, caspase-3 activation, and amyloid β1-42-induced cell death, also suppressing mitogen-activated protein kinase kinase 4 (MKK4) and c-jun N-terminal kinase (JNK) signaling activated by n |
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DCC4233 |
Pqc-078 |
Novel inhibitor of IMPDH enzyme |
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DCC4234 |
Pqq-tme |
Novel human double minute 2 (HDM2) inhibitor |
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DCC4235 |
Pqsr Antagonist M64 |
Quorum sensing modulator as a PqsR antagonist |
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DCC4236 |
Pradigastat
Featured
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Pradigastat (LCQ-908) is a potent, selective and orally active diacylglycerol acyltransferase 1 (DGAT1) inhibitor. Pradigastat has anti-obesity and anti-diabetic effects. |
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DCC4237 |
Pravadoline Maleate |
Inhibitor of prostaglandin (PG) synthesis |
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DCC4238 |
Prazosin |
Inverse agonist at alpha-1 adrenergic receptors |
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DCC4239 |
Prexasertib Monolactate Monohydrate |
Novel inhibitor of checkpoint kinase 1 (CHK1) |
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DCC4240 |
Pridopidine Hydrochloride |
Inducer of Functional Neurorestoration Via the Sigma-1 Receptor |
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DCC4241 |
prmt3 Inhibitor 1 |
Allosteric inhibitor of protein arginine methyltransferase 3 (PRMT3) |
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DCC4242 |
prmt3 Inhibitor 14u |
Potent and selective inhibitor of protein arginine methyltransferase 3 (PRMT3) |
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DCC4243 |
Prmt4-in-1 |
Novel potent and selective inhibitor of PRMT4 (also known as CARM1) |
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DCC4244 |
Prmt5-in-4b14 |
Novel potent PRMT5 inhibitor, exhibiting potent anti-proliferative activity against a panel of leukemia and lymphoma cells |
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DCC4245 |
Prmt5-in-c17
Featured
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Novel potent, selective, and cell active protein arginine methyltransferase 5 (PRMT5) inhibitor |
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DCC4246 |
Prmts Inhibitor A36 |
Potent inhibitor of protein arginine methyltransferases (PRMTs) |
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DCC4247 |
Prmts Inhibitor A9 |
Potent inhibitor of protein arginine methyltransferases (PRMTs) |
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DCC4248 |
Prn1008 |
Novel, Reversible Covalent BTK Inhibitor for Rheumatoid Arthritis |
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DCC4249 |
Prn1126 |
Novel reversible covalent selective LMP7 inhibitor |
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DCC4250 |
pr-nhp5g |
Antagonist at the NR1/NR2A subtype but an agonist at the NR1/NR2D subtype |
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DCC4251 |
Probimane |
Potent inhibitor of tumor metastasis, inhibiting calmodulin, sialic acid, lipoperoxidation, fibrinogen, cell-movement and the cell-cycle arrest |
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DCC4252 |
Procaspase-8 Inhibitor 63-r |
Novel selective procaspase-8 (Pro-C8) Inhibitor covalently binding the zymogen, or inactive precursor (pro-form), of caspase-8, but not other caspases |
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DCC4253 |
Pro-nbdhex |
Prodrug of NBDHEX, selectively inhibiting glutathione transferase (GST P1-1) with better water solubility, and more potent anticancer activities |
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DCC4254 |
Protac 14a |
Novel potent cereblon degrader with DC50 of 200 nM, and 64% protein degradation, as quantified by western blot |
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DCC4256 |
Protac Cp17 |
Novel highly potent degrader against EGFRL858R/T790M and EGFRdel19, reaching the lowest DC 50 values among all reported EGFR-targeting PROTACs |
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