DCC4466 |
Ro5234444 |
Orally active chemokine receptor CCR2 antagonist preventing glomerulosclerosis and renal failure in type 2 diabetes |
|
DCC4467 |
Ro5527239 |
Novel potent, orally available GPBAR1 agonist |
|
DCC4468 |
Ro-57-bpyne |
Novel γ-secretase modulator photoaffinity probe, identifying distinct allosteric binding sites on presenilin that can be exploited to reduce levels of pathogenic Aβ species |
|
DCC4469 |
Ro6800020 |
Potent γ-secretase modulator (GSM) |
|
DCC4470 |
Ro6842262 |
Novel potent and selectve LPA1 antagonist, attenuating NHLF human lung fibroblast cell proliferation and contraction in vitro, reducing plasma histamine levels in mouse LPA-challenge model |
|
DCC4471 |
Ro7101556 |
Novel potent γ-secretase modulator (GSM) with high solubility, balanced lipophilicity, and showing no phototoxicity and PIK4CB side bing activity |
|
DCC4472 |
Robalzotan |
Selective antagonist at the 5-HT1A receptor |
|
DCC4473 |
Rocepafant |
Platelet-activating factor (PAF-R) antagonist, selectively for intracellular PAF binding sites |
|
DCC4474 |
Rockii-in-di |
Novel potent competitive inhibitor of Rho-associated coiled-coil-containing protein kinase 2 (ROCKII) |
|
DCC4475 |
Rock-in-(r)14f |
Novel potent ROCK inhibitor |
|
DCC4476 |
Rock-in-32 |
Potent Rho--kinase (ROCK) inhibitor |
|
DCC4477 |
Rock-in-d1 |
Novel potent and selective ROCK inhibitor |
|
DCC4478 |
Rock-in-d2 |
Novel potent and selective ROCK inhibitor |
|
DCC4479 |
Rock-in-d3 |
Novel potent and selective ROCK inhibitor |
|
DCC4480 |
Rohitukine |
Anti-cancer agent, acting through gastrin antagonism and H /K -ATPase inhibition, modulating apoptosis pathways, antidyslipidemic, antiadipogenic, gastroprotective, antifertility, and antileishmanial |
|
DCC4481 |
Ronifibrate |
Lipid modifying agent; Antihyperlipidemic and antiarteriosclerotic |
|
DCC4482 |
Rooperol |
Novel p38α kinase inhibitor; Antioxidant |
|
DCC4483 |
Ropizine |
Allosteric modulator of dextromethorphan binding to high-affinity sigma receptors |
|
DCC4484 |
Ror Modulator I |
The first potent inverse agonist of retinoid-related orphan receptor (ROR) with dual selectivity for RORβ and RORγt |
|
DCC4485 |
Rorgammat Agonist 8-074 |
Novel potent and selective RORγt agonist, showing robust antitumor efficacy in syngeneic tumor models and improving the efficacy of anti‑PD‑1 in a murine lung cancer model |
|
DCC4486 |
Rorgammat Inhibitor I |
Novel RORgammaT inhibitor |
|
DCC4487 |
Rorγt Agonist |
Novel RORγt agonist |
|
DCC4488 |
Rorγt-inverse-agonist-1j |
Novel potent RORγt inverse agonist |
|
DCC4489 |
Rosma-18-d6 |
Novel potent and selective CB2 probe (Ki for CB2: 0.8 nM and >12000 selectivity over CB1) |
|
DCC4490 |
Ros-modulator-3b |
Novel P2X3 antagonist |
|
DCC4491 |
Rostaporfin |
Photosensitiser for the treatment of age-related macular degeneration |
|
DCC4492 |
Rovafovir |
Novel nucleoside phosphonate HIV reverse transcriptase (RT) inhibitor |
|
DCC4493 |
Rovafovir Etalafenamide |
Prodrug of the novel nucleoside phosphonate HIV reverse transcriptase (RT) inhibitor GS-9148 |
|
DCC4494 |
Roxatidine Acetate |
Specific and competitive H2 receptor antagonist |
|
DCC4495 |
Rp-001 Hydrochloride |
Potent agonist of S1P1 receptors |
|