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Cat. No. Product name CAS No.
DC10686 Cosan-528 Featured

Cosan-528 is a bioactive chemical.

96686-51-0
DC9554 Cot inhibitor-1

Cot inhibitor-1 is a COT/Tpl2 inhibitor.

915365-57-0
DC20933 Cotylimide-VI

Cotylimide-VI (CTL-VI) is a small molecule that perturbs plant hormone strigolactone accumulation and inhibits hypocotyl growth..

419539-64-3
DC10363 Coumestrol Featured

Coumestrol, a phytoestrogen present in soybean products, exhibits activities against cancers, neurological disorders, and autoimmune diseases. It suppresses proliferation of ES2 cells with an IC50 of 50 μM.

479-13-0
DC21413 Cowanin

Cowanin is a novel natural product from Garcinia speciosa that inhibits the Notch signaling pathway with IC50 of 2.4 uM.

21044-85-9
DC12046 CP 105696 Featured

CP-105696 is a potent and selective Leukotriene B4 Receptor antagonist, with an IC50 of 8.42 nM.

158081-99-3
DC23320 CP 31398 dihydrochloride Featured

CP-31398 is a small molecule p53 reactivator that protects p53 from thermal denaturation, not only reactivates mutant p53 but also induces stabilization of wild type p53.

1217195-61-3
DC23610 CP-339818 hydrochloride Featured

CP-339818 is a potent, selective, non-peptide KV1.3 channel antagonist with IC50 of 200 nM.

478341-55-8
DC23415 CP-481715

CP-481715 is a potent and selective CCR1 antagonist with Ki of 9.2 nM and IC50 of 74 nM, lacks intrinsic agonist activity and .

212790-31-3
DC9265 CP-640186 hydrochloride Featured

CP-640186 Hcl is an isozyme-nonselective acetyl-CoA carboxylase (ACC) inhibitor with IC50s of 53 nM and 61 nM for rat liver ACC1 and rat skeletal muscle ACC2 respectively; with improved metabolic stability vs CP-610431.

591778-70-0
DC7975 CP 640186 Featured

CP-640186 is an isozyme-nonselective acetyl-CoA carboxylase inhibitor with IC50s of 53 nM and 61 nM for rat liver ACC1 and rat skeletal muscle ACC2 respectively.

591778-68-6
DC11410 CP-671305 Featured

CP-671305 is a potent and selective inhibitor of phosphodiesterase 4.

445295-04-5
DC8251 CP-724,714

CP-724,714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >640-fold selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc. Phase 2.

383432-38-0
DC23544 CPG-52364

CPG-52364 (CPG52364) is an orally available, small molecule TLR7/8/9 antagonist for the treatment of systemic lupus erythematosus and other autoimmune disorders..

1093135-60-4
DC10506 CPHPC(Miridesap) Featured

CPHPC(GSK2315698,Miridesap) is a divalent crosslinker of SAP that causes rapid depletion of circulating SAP via hepatic clearance.

224624-80-0
DC7564 CPI 0610(Pelabresib) Featured

CPI 0610 is a potent, selective, and cell-active BET bromodomain inhibitor with IC50 of 39 nM for BRD4-BD1 in TR-FRET assay.

1845726-14-8
DC9736 CPI1189(REN-1189) Featured

CPI-1189 prevents apoptosis and reduces glial fibrillary acidic protein immunostaining in a TNF-alpha infusion model for AIDS dementia complex.

183619-38-7
DC8001 CPI 169 R-enantiomer Featured

CPI-169 R is a novel and potent EZH2 inhibitor with IC50 <1 nM(inhibition of the catalytic activity of PRC2.

DC8466 CPI-169 (racemate) Featured

CPI-169 racemate is the racemate form of CPI-169, which is a novel and potent EZH2 inhibitor with IC50 <1 nM(inhibition of the catalytic activity of PRC2); decreases cellular levels of H3K27me3 with an EC50 of 70 nM, and triggers cell cycle arrest and apo

1450655-76-1
DC8002 CPI-360 (R) Featured

CPI-360 is a compound in design and preparation of wew palladium precatalysts for C-C and C-N cross-coupling reactions.

1802175-06-9
DC10593 CPI-455 analogue(KDM5 inhibitor) Featured

CPI-455 analogue is a selective inhibitor of KDM5 demethylases.

DC10591 CPI-613 Featured

CPI-613 is an E1α pyruvate dehydrogenase (PDH) modulator that prevents cancer cells from metabolizing glucose for energy. CPI-613 has been granted orphan drug status by the US FDA for pancreatic cancer.

95809-78-2
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