DCC5096 |
Texasin |
Potent and selective human leukocyte 5-lipoxygenase (5-LOX) inhibitor |
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DCC5097 |
Tezosentan |
Novel endothelin (ET) receptor antagonist |
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DCC5098 |
Tfah-10n |
Novel multipotent anti-Alzheimer agent, selectively inhibiting human butyrylcholinesterase (BChE), having strong antioxidant activity and good β-amyloid (Aβ) anti-aggregation properties |
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DCC5099 |
Tfgf-18 |
Novel GSK-3β inhibitor, showing anti-neuroinflammatory effects in lipopolysaccharide (LPS) activation of spontaneously immortalized SIM-A9 microglial cells and of mouse cortical microglia, inhibiting LPS-induced production of nitric oxide and the proinfla |
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DCC5100 |
Tfmo-1 |
Novel cell-active, selective class IIa HDAC inhibitor |
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DCC5101 |
Tfmo-12 |
CNS-penetrant selective class IIa histone deacetylase (HDAC) inhibitor, exploiting the >100-fold selectivity over class I/IIb HDACs |
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DCC5102 |
Tfr4oht |
Cyclized tamoxifen analog, selective ER modulator (SERM) |
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DCC5103 |
Tg-0054 |
Novel and Potent Stem Cell Mobilizer; Inhibitor of SDF-1α/CXCR4 binding |
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DCC5104 |
Tg-0205221 |
Novel potent SARS coronavirus (CoV) 3CL protease inhibitor (Ki = 53 nM) |
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DCC5105 |
Tg100948 |
Novel dual VEGFR/Src kinase inhibitor |
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DCC5106 |
Tg101114 |
Novel inhibitor of T315I mutant enzyme, exhibiting reasonable in vivo efficacy in a xenograft mouse model harboring T315I |
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DCC5107 |
Tg11-77 Hydrochloride |
Novel, Potent, Selective, Water Soluble, Brain-Permeable EP2 Receptor Antagonist |
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DCC5108 |
Tg-2112x |
Novel inhibitor of mitochondrial calcium uptake (#333333; font-family: "Open Sans", HelveticaNeue, "Helvetica Neue", Helvetica, Arial, sans-serif; font-size: 15px; font-style: normal; font-variant-ligatures: normal; font-variant-caps: normal; font-weight: |
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DCC5109 |
Tg2-in-3h |
Highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (TG2) inhibitor |
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DCC5110 |
Tg3-95-1 |
EP2 allosteric potentiator |
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DCC5111 |
Tg4-166 |
Potent and selective nociceptin opioid receptor (NOP) agonist |
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DCC5112 |
tg4-290-1 |
Potent and selective nociceptin opioid receptor (NOP) agonist |
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DCC5113 |
tg4-292-1 |
Potent and selective nociceptin opioid receptor (NOP) agonist |
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DCC5114 |
Tg4-294-2 |
Potent and Selective Antagonist for Human EP2 Receptors |
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DCC5115 |
Tgp-200c |
Novel potent and structure-specific inhibitor of pre-miR-200c, reversing a type 2 diabetes phenotype |
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DCC5116 |
Tgr5 Agonist 11d-na |
Novel potent TGR5 agonist, displayind a significant glucose-lowering effect and stimulated GLP-1 and insulin secretion in TGR5H88Y mice but not in wild-type animals |
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DCC5117 |
Tgr5-agonist-17 |
Novel Potent Agonist of TGR5 Receptor |
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DCC5118 |
Tgx-115 |
Cell-permeable, potent, and selective inhibitor of PI 3-K isoforms p110ß/p110d |
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DCC5119 |
Tgx-155 |
Potent and selective inhibitor of PI 3-K |
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DCC5120 |
Th1027 |
Novel highly potent and specific inhibitor of TLR8, targeting an unconventional pocket on the TLR8 protein-protein Interface |
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DCC5121 |
Thaigranatin T |
Natural potent human carboxylesterase 2 (hCES2) inhibitor (IC50: 5.05 μM) |
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DCC5122 |
Thalassosamide |
Natural antibiotic, being active against P. aeruginosa both in vitro and in vivo. |
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DCC5123 |
Thdp-17 |
Novel glutaminase activity inhibitor, showing a partial uncompetitive inhibition in vitro and a significant reduction of ammonia and glutamate production in vivo |
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DCC5124 |
Thiamphenicol Palmitate |
Prodrug of Thiamphenicol, inhibiting the 50S subunit of the bacterial ribosome and protein translation |
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DCC5125 |
Thiazolidinedione-8 |
Novel antibiofilm agent, disturbing symbiotic balance between C. albicans and S. mutans in dual species biofilm |
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