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AMG PERK 44

  Cat. No.:  DC28501  
Chemical Structure
1883548-84-2
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Field of application
AMG PERK 44 is an orally active and highly selective PERK inhibitor with an IC50 of 6 nM. AMG PERK 44 has 1000-fold and 160-fold selectivity over GCN2 (IC50=7300 nM) and B-Raf (IC50 >1000 nM), respectively.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1883548-84-2
Formula: C34H29ClN4O2
M.Wt: 561.07
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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MSDS_12554_DC28501_1883548-84-2
COA
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Cat. No. Product name Field of application
DC41027 MK-28 MK-28 is a potent and selective PERK activator. MK-28 exhibits remarkable pharmacokinetic properties and high BBB penetration in mice.
DC28778 PERK-IN-2 PERK-IN-2 is a potent PERK inhibitor with an IC50 of 0.2 nM.
DC28683 PERK-IN-3 PERK-IN-3 is a potent PERK inhibitor with an IC50 of 7.4 nM.
DC28501 AMG PERK 44 AMG PERK 44 is an orally active and highly selective PERK inhibitor with an IC50 of 6 nM. AMG PERK 44 has 1000-fold and 160-fold selectivity over GCN2 (IC50=7300 nM) and B-Raf (IC50 >1000 nM), respectively.
DC12283 CCT020312 CCT020312 is capable of delivering potent, and eukaryotic initiation factor 2-alpha kinase 3 (EIF2AK3) selective, proliferation control and also is an activator of RNA-like endoplasmic reticulum kinase (PERK).
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