PERK-IN-3

  Cat. No.:  DC28683  
Chemical Structure
1337532-08-7
For research use only. We do not sell to patients.
We match the best price and quality on market.
Email:order@dcchemicals.com  sales@dcchemicals.com
Tel:+86-021-58447131
We are official vendor of:
  • 20
  • 19
  • 18
  • 17
  • 16
  • 15
  • 14
  • 12
  • 11
  • 10
  • 9
  • 8
  • 13
  • 6
  • 5
  • 4
  • 3
  • 2
  • 1
More than 5000 active chemicals with high quality for research!
Field of application
PERK-IN-3 is a potent PERK inhibitor with an IC50 of 7.4 nM.
Cas No.: 1337532-08-7
Formula: C22H16F2N4O2
M.Wt: 406.38
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
TITLE DOWNLOAD
MSDS_12735_DC28683_1337532-08-7
COA
LOT NO. DOWNLOAD
Cat. No. Product name Field of application
DC41027 MK-28 MK-28 is a potent and selective PERK activator. MK-28 exhibits remarkable pharmacokinetic properties and high BBB penetration in mice.
DC28778 PERK-IN-2 PERK-IN-2 is a potent PERK inhibitor with an IC50 of 0.2 nM.
DC28683 PERK-IN-3 PERK-IN-3 is a potent PERK inhibitor with an IC50 of 7.4 nM.
DC28501 AMG PERK 44 AMG PERK 44 is an orally active and highly selective PERK inhibitor with an IC50 of 6 nM. AMG PERK 44 has 1000-fold and 160-fold selectivity over GCN2 (IC50=7300 nM) and B-Raf (IC50 >1000 nM), respectively.
DC12283 CCT020312 CCT020312 is capable of delivering potent, and eukaryotic initiation factor 2-alpha kinase 3 (EIF2AK3) selective, proliferation control and also is an activator of RNA-like endoplasmic reticulum kinase (PERK).
X