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Home > Inhibitors & Agonists > Cytoskeleton/Cell Adhesion Molecules > Integrin

Cyclo(RGDyK)

  Cat. No.:  DC8399   Featured
Chemical Structure
250612-42-1
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More than 5000 active chemicals with high quality for research!
Field of application
Cyclo(RGDyK) is a potent and selective αVβ3 integrin inhibitor with IC50 of 20 nM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 250612-42-1
Chemical Name: Cyclo(RGDyK) trifluoroacetate
Synonyms: Cyclic Arg-Gly-Asp-D-Tyr-Lys;Cyclo(RGDyK);AK685805;Cyclo(RGDyK) trifluoroacetate
SMILES: FC(C(=O)O)(F)F.FC(C(=O)O)(F)F.O=C1C(CCCCN)NC(C(CC2C=CC(=CC=2)O)NC(C(CC(=O)O)NC(CNC(C(CCC/N=C(\N)/N)N1)=O)=O)=O)=O
Formula: C31H43F6N9O12
M.Wt: 847.716648340225
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Cyclo(RGDyK) trifluoroacetate is a potent and selective αVβ3 integrin inhibitor with an IC50 of 20 nM.
In Vitro: Cyclo(RGDyK) (c(RGDyK(SAA)) shows high affinity and selectivity for αVβ3 over αVβ5 (IC50=4000 nM) and αIIbβ3 (IC50=3000 nM)[1].
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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