| Cas No.: | |
| Chemical Name: | 5-((3S,4R)-3-(((1H-indazol-5-yl)oxy)methyl)piperidin-4-yl)-N-((1H-pyrazol-5-yl)methyl)-2-fluorobenzamide |
| Synonyms: | CCG258748;CCG-258748 |
| SMILES: | C(NCC1NN=CC=1)(=O)C1=CC([C@H]2CCNC[C@@H]2COC2C=CC3=C(C=2)C=NN3)=CC=C1F |
| Purity: | >98% |
| Sotrage: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
| Description: | A potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM; displays 30-fold selectivity over GRK5, and no significant inhibitory activity against GRK1, PKA and ROCK1. |
MSDS
COA
| LOT NO. | DOWNLOAD |
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| 2018-0101 |
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