CCG 258001

  Cat. No.:  DC11958  
Chemical Structure
2055990-96-8
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More than 5000 active chemicals with high quality for research!
Field of application
A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM.
Cas No.: 2055990-96-8
Chemical Name: 5-(((3S,4R)-4-(4-fluorophenyl)-1-methylpiperidin-3-yl)methoxy)-1H-indazole
Synonyms: CCG258001;CCG-258001
SMILES: N1C2=C(C=C(OC[C@@H]3[C@@H](C4=CC=C(F)C=C4)CCN(C)C3)C=C2)C=N1
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM; displays >100-fold selectivity over GRK5, GRK1, PKA and ROCK1.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
DC11956 CCG 258748 A potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.
DC11957 CCG 224061 A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 66 nM.
DC11958 CCG 258001 A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM.
DC11765 GRK2-IN-115h hydrochloride A highly potent and selective GRK2 inhibitor with IC50 of 18 nM.
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