Cas No.: | 2055990-96-8 |
Chemical Name: | 5-(((3S,4R)-4-(4-fluorophenyl)-1-methylpiperidin-3-yl)methoxy)-1H-indazole |
Synonyms: | CCG258001;CCG-258001 |
SMILES: | N1C2=C(C=C(OC[C@@H]3[C@@H](C4=CC=C(F)C=C4)CCN(C)C3)C=C2)C=N1 |
Purity: | >98% |
Sotrage: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Description: | A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM; displays >100-fold selectivity over GRK5, GRK1, PKA and ROCK1. |