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IHMT-PI3Kδ-372

  Cat. No.:  DC42415   Featured
Chemical Structure
2429889-62-1
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More than 5000 active chemicals with high quality for research!
Field of application
IHMT-PI3Kδ-372 is a potent and selective PI3Kδ with an IC50 of 14 nM. IHMT-PI3Kδ-372 shows high selectivity over other class I PI3Ks (56∼83 fold) and other protein kinases. IHMT-PI3Kδ-372 can be uesd for chronic obstructive pulmonary disease (COPD) research.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2429889-62-1
Chemical Name: Ihmt-PI3K|A-372
Synonyms: IHMT-PI3K;Ihmt-PI3K|A-372
SMILES: FC1=C([H])C([H])=C([H])C2=C1C(N(C([C@@]([H])(C([H])([H])C([H])([H])[H])N1C3C(=C(N([H])[H])N=C([H])N=3)C(C3C([H])=C([H])C(=C(C=3[H])F)OC([H])([H])[H])=N1)=N2)C1([H])C([H])([H])C1([H])[H])=O
Formula: C26H23F2N7O2
M.Wt: 503.5033
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
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MSDS_26022_DC42415_2429889-62-1
COA
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Cat. No. Product name Field of application
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DC72848 Leniolisib phosphate Leniolisib (CDZ173) phosphate is a potent and selective PI3Kδ inhibitor. Leniolisib phosphate has the potential for immunodeficiency disorders treatment.
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DC42415 IHMT-PI3Kδ-372 IHMT-PI3Kδ-372 is a potent and selective PI3Kδ with an IC50 of 14 nM. IHMT-PI3Kδ-372 shows high selectivity over other class I PI3Ks (56∼83 fold) and other protein kinases. IHMT-PI3Kδ-372 can be uesd for chronic obstructive pulmonary disease (COPD) research.
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DC40777 MSC2360844(IOA-244 /roginolisib) MSC2360844 is a potent, orally active and selective PI3Kδ inhibitor, with an IC50 of 145 nM. MSC2360844 shows highly selective against a panel of 278 additional kinases.
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