LPA2 antagonist 2

  Cat. No.:  DC28324  
Chemical Structure
36840-10-5
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More than 5000 active chemicals with high quality for research!
Field of application
LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM, which is >480-fold more selective than LPA3 (IC50 of 13.85 μM).
Cas No.: 36840-10-5
Formula: C20H16N2O6
M.Wt: 380.35
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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DC42560 1-Oleoyl lysophosphatidic acid 1-Oleoyl lysophosphatidic acid (1-Oleoyl-sn-glycero-3-phosphate) is an abundant LPA species with high biological activity due to its strong affinity for the LPA receptors. 1-Oleoyl lysophosphatidic acid is commonly used in most laboratories as a reagent for LPA receptor activation. 1-Oleoyl lysophosphatidic acid increases SRE-drivenβ-galactosidase activity.
DC28324 LPA2 antagonist 2 LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM, which is >480-fold more selective than LPA3 (IC50 of 13.85 μM).
DC28232 CYM50260 CYM50260 is a potent and exquisitely selective sphingosine-1-phosphate 4 receptor (S1P4-R) agonist with an EC50 of 45 nM. CYM50260 displays no activity against S1P1-R, S1P2-R, S1P3-R and S1P5-R.
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DC8621 AM095 AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.
DC11561 SPM-242 racemate A potent, selective S1P3 antagonist with Ki of 0.25 nM.
DC11560 SPM-242 A potent, selective S1P3 antagonist with Ki of 0.25 nM.
DC11605 ONO-0300302 A novel potent, slow tight binding LPA1 receptor antagonist with IC50 of 86 nM, Kd of 0.34 nM.
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