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SSD114 hydrochloride

  Cat. No.:  DC10651   Featured
Chemical Structure
2319790-02-6
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More than 5000 active chemicals with high quality for research!
Field of application
SSD114 is a novel GABAB positive allosteric modulator.
Cas No.: 2319790-02-6
Chemical Name: SSD114 hydrochloride
Synonyms: SSD-114,SSD 114
SMILES: FC(F)(F)C1C=CC(C2N=C(NC3CCCCC3)N=C(OC)C=2)=CC=1.[H]Cl
Formula: C18H21ClF3N3O
M.Wt: 387.83
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: SSD114 is a novel GABAB positive allosteric modulator. SSD114 potentiates the GABA inhibition of adenylyl-cyclase mediated by GABAB receptors. SSD114 is also effective in vivo potentiating baclofen-induced sedation/hypnosis in mice, with no effect when tested alone. These findings indicate that SSD114, a molecule with a different chemical structure compared to known GABAB PAMs, is a novel GABAB PAM with potential usefulness in the GABAB-receptor research field.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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