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Vps34-IN-1

  Cat. No.:  DC8650   Featured
Chemical Structure
1383716-33-3
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More than 5000 active chemicals with high quality for research!
Field of application
VPS34-IN1 is a potent and highly selective Vps34 inhibitor with IC50 of 25 nM invitro,which does not significantly inhibit the isoforms of class I as well as class II PI3Ks.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1383716-33-3
SMILES: CC(C)(O)CNC1=NC=C(C2=CC=NC(NC3=CC=NC(Cl)=C3)=N2)C(CC4CC4)=N1
Formula: C21H24ClN7O
M.Wt: 425.91
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Vps34-IN-1 is an inhibitor of Vps34 extracted from patent WO2012085815A1, compound example 16a, with an IC50 of 4 nM.
Target: Vps34:4 nM (IC50)
References: [1]. WO/2012085815 A1
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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