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ALK5-IN-9

  Cat. No.:  DC50283  
Chemical Structure
2489611-06-3
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More than 5000 active chemicals with high quality for research!
Field of application
ALK5-IN-9 (Compound 8h) is a potent and orally active inhibitor of TGFβRI (ALK5). ALK5-IN-9 inhibits ALK5 autophosphorylation and NIH3T3 cell activity with IC50 values of 25 nM and 74.6 nM, respectively. ALK5-IN-9 also shows favorable pharmacokinetic profile and ameliorated hERG inhibition. ALK5-IN-9 has the potential for the research of cancer disease.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2489611-06-3
Chemical Name: ALK5-IN-9
Formula: C29H35F3N6O3
M.Wt: 572.62
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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