PCLX-001

  Cat. No.:  DC71735   Featured
Chemical Structure
1215011-08-7
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Field of application
PCLX-001 is an orally acitve, small-molecule, dual N-myristoyltransferase (NMT) inhibitor, with IC50s of 5 nM (NMT1) and 8 nM (NMT2), respectively.
Cas No.: 1215011-08-7
Chemical Name: 2,6-Dichloro-4-(2-Piperazin-1-Ylpyridin-4-Yl)-N-(1,5-Dimethyl,3-Isobutyl-1h-Pyrazol-4-Yl)benzenesulfonamide
Synonyms: 2,6-Dichloro-4-(2-Piperazin-1-Ylpyridin-4-Yl)-N-(1,5-Dimethyl,3-Isobutyl-1h-Pyrazol-4-Yl)benzenesulfonamide;2,6-Dichloro-N-(3-isobutyl-1,5-dimethyl-1H-pyrazol-4-yl)-4-(2-(piperazin-1-yl)pyridin-4-yl)benzenesulfonamide;starbld0016320;5HY8BYC3Q6;BDBM184902;BDBM50033418;DDD 86481;US9156811, DDD86481;Q27464265;2,6-Dichloro-N-[1,5-dimethyl-3-(2-methylpropyl)-1H-pyrazol-4-yl]-4-[2-(1-piperazinyl)-4-pyridinyl]benz
SMILES: ClC1C([H])=C(C([H])=C(C=1S(N([H])C1=C(C([H])([H])[H])N(C([H])([H])[H])N=C1C([H])([H])C([H])(C([H])([H])[H])C([H])([H])[H])(=O)=O)Cl)C1C([H])=C([H])N=C(C=1[H])N1C([H])([H])C([H])([H])N([H])C([H])([H])C1([H])[H]
Formula: C24H30Cl2N6O2S
M.Wt: 537.5050
Purity: 98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
DC71735 PCLX-001 PCLX-001 is an orally acitve, small-molecule, dual N-myristoyltransferase (NMT) inhibitor, with IC50s of 5 nM (NMT1) and 8 nM (NMT2), respectively.
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