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Umbralisib tosylate

  Cat. No.:  DC71904  
Chemical Structure
1532533-72-4
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More than 5000 active chemicals with high quality for research!
Field of application
Umbralisib (TGR-1202) tosylate is an orally active, potent and selective dual PI3Kδ and casein kinase-1-ε (CK1ε) inhibitor, with EC50 of 22.2 nM and 6.0 μM, respectively. Umbralisib tosylate exhibits unique immunomodulatory effects on chronic lymphocytic leukemia (CLL) T cells. Umbralisib tosylate can be used for haematological malignancies reseach.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1532533-72-4
Chemical Name: Umbralisib tosylate
SMILES: O=C1C(C2=CC=CC(F)=C2)=C([C@@H](N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)C)OC6=CC=C(F)C=C16.O=S(C7=CC=C(C)C=C7)(O)=O
Formula: C38H32F3N5O6S
M.Wt: 743.75
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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