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Cat. No. Product name CAS No.
DC8487 Gemcitabine elaidate Featured

Gemcitabine elaidate is a lipophilic, unsaturated fatty acid ester derivative of gemcitabine (dFdC), an antimetabolite deoxynucleoside analogue, with potential antineoplastic activity.

210829-30-4
DC2107 Gemcitabine HCl (Gemzar,LY188011) Featured

Gemcitabine Hydrochloride (Gemzar) is a DNA synthesis inhibitor with IC50 of 50 nM, 40 nM, 18 nM and 12 nM in PANC1, MIAPaCa2, BxPC3 and Capan2 cells, respectively,showed potent activity against COVID-19(SARS-COV-2) with EC50 MERS-COV(1.216), SARS-COV(4.9

122111-03-9
DC10590 Gemcitabine monophosphate Featured

Gemcitabine monophosphate disodium salt, also called GemMP, is a monophosphate derivative of Gemcitabine.

1638288-31-9
DC3159 Gemifioxacin Featured

Gemifloxacin mesylate (trade name Factive, Oscient Pharmaceuticals) is an oral broad-spectrum quinolone antibacterial agent used in the treatment of acute bacterial exacerbation of chronic bronchitis and mild-to-moderate pneumonia.

210353-53-0
DC2092 Genistein Featured

Genistein is a highly specific inhibitor of protein tyrosine kinase (PTK).

446-72-0
DC2093 Genistin Featured

Genistin is an isoflavone glycoside found in soy-based products. Can be used as a negative control for the PTK inhibitor Genistein

529-59-9
DCAPI1064 mixtures of three isomers (Gentamicins C1, C2, and C1(subA). Featured

Gentamycin sulfate (Gentacycol)

1405-41-0
DC7417 Genz-123346 Featured

Genz-123346 free base is an inhibitor of GL1 synthase that blocks the conversion of ceramide to GL1; IC50 for GM1 inhibition is 14 nM.

491833-30-8
DC10161 Gepotidacin Featured

Gepotidacin (GSK2140944) is a novel triazaacenaphthylene bacterial type II topoisomerase inhibitor.

1075236-89-3
DC7132 GF 109203X Featured

GF109203X is a potent PKC inhibitor with IC50 of 20 nM, 17 nM, 16 nM, and 20 nM for PKCα, PKCβI, PKCβII, and PKCγ, respectively, showing more than 3000-fold selectivity for PKC as compared to EGFR, PDGFR and insulin receptor.

133052-90-1
DC21043 GGTI 2417 Featured

GGTI 2417 is the methyl ester prodrug of GGTI-2418, a highly potent, competitive, and selective inhibitor of GGTase I.

501010-05-5
DC21044 GGTI 2418 Featured

GGTI 2418 (PTX 100) is a highly potent, competitive, and selective peptidomimetic inhibitor of geranylgeranyltransferase I (GGTI) with IC50 of 9.5 nM, displays 5,600-fold selectivity over FTase.

501010-06-6
DC21042 GGTI-2147 Featured

GGTI-2147 is a non-thiol peptidomimetic that inhibits GGTase I and blocks geranyl-geranylation of Rap1A (IC50=0.5 uM).

191102-87-1
DC11246 Ghrelin agonist HM01 Featured

Ghrelin agonist HM01 is a novel potent, orally available ghrelin (GHS-R) agonist with Ki of 1.42 nM (human GHS-R1a), induces potent activation of intracellular calcium signaling with EC50 of 1.25 nM.

1394860-28-6
DC10883 GI254023X Featured

GI254023X is a potent MMP9 and ADAM10 inhibitor with IC50s of 2.5 and 5.3 nM, respectively.

260264-93-5
DC10490 GIBH-130 Featured

GIBH-130 is a novel inhibitor of neuroinflammation effective in Alzheimer’s disease models.

1252608-59-5
DC7432 Givinostat (ITF2357) Featured

Givinostat (ITF2357) is a potent HDAC inhibitor for maize HD2, HD1B and HD1A with IC50 of 10 nM, 7.5 nM and 16 nM. Phase 1/2.

732302-99-7
DC10081 GJ103 Featured

GJ103 is an active analog of the read-through compound GJ072.

1459687-89-8
DC10080 GJ103 (sodium salt) Featured

GJ103 sodium salt is an active analog of the read-through compound GJ072.

1459687-96-7
DC9855 GK921 Featured

GK921 is a transglutaminase 2 (TGase 2) inhibitor with average GI50 of 0.9 uM in cancer cell lines.

1025015-40-0
DC8118 GKT137831(Setanaxib) Featured

GKT137831 is a novel and specific dual Nox1/Nox4 inhibitor with Ki of 140±40 nM and 110±30 nM; a potent inhibitor of fibrosis and hepatocyte apoptosis.

1218942-37-0
DC21049 Glabrescione B Featured

Glabrescione B (GlaB) is a small molecule binding to Gli1 zinc finger and impairing Gli1 activity by interfering with Gli1/DNA interaction, inhibits Hh signaling by impairing Gli1 function; inhibits the growth of Hedgehog-dependent tumor cells in vitro and in vivo, inhibits Gli1-dependent growth of cerebellum-derived normal progenitors; inhibits the growth of Gli-dependent medulloblastoma and tumor-derived stem-like cells; inhibits the growth of Gli-dependent basal cell carcinoma in vitro and in vivo.

65893-94-9
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