Cat. No. | Product name | CAS No. |
DC8487 |
Gemcitabine elaidate
Featured
Gemcitabine elaidate is a lipophilic, unsaturated fatty acid ester derivative of gemcitabine (dFdC), an antimetabolite deoxynucleoside analogue, with potential antineoplastic activity. |
210829-30-4 |
DC2107 |
Gemcitabine HCl (Gemzar,LY188011)
Featured
Gemcitabine Hydrochloride (Gemzar) is a DNA synthesis inhibitor with IC50 of 50 nM, 40 nM, 18 nM and 12 nM in PANC1, MIAPaCa2, BxPC3 and Capan2 cells, respectively,showed potent activity against COVID-19(SARS-COV-2) with EC50 MERS-COV(1.216), SARS-COV(4.9 |
122111-03-9 |
DC10590 |
Gemcitabine monophosphate
Featured
Gemcitabine monophosphate disodium salt, also called GemMP, is a monophosphate derivative of Gemcitabine. |
1638288-31-9 |
DC3159 |
Gemifioxacin
Featured
Gemifloxacin mesylate (trade name Factive, Oscient Pharmaceuticals) is an oral broad-spectrum quinolone antibacterial agent used in the treatment of acute bacterial exacerbation of chronic bronchitis and mild-to-moderate pneumonia. |
210353-53-0 |
DC2092 |
Genistein
Featured
Genistein is a highly specific inhibitor of protein tyrosine kinase (PTK). |
446-72-0 |
DC2093 |
Genistin
Featured
Genistin is an isoflavone glycoside found in soy-based products. Can be used as a negative control for the PTK inhibitor Genistein |
529-59-9 |
DCAPI1064 |
mixtures of three isomers (Gentamicins C1, C2, and C1(subA).
Featured
Gentamycin sulfate (Gentacycol) |
1405-41-0 |
DC7417 |
Genz-123346
Featured
Genz-123346 free base is an inhibitor of GL1 synthase that blocks the conversion of ceramide to GL1; IC50 for GM1 inhibition is 14 nM. |
491833-30-8 |
DC10161 |
Gepotidacin
Featured
Gepotidacin (GSK2140944) is a novel triazaacenaphthylene bacterial type II topoisomerase inhibitor. |
1075236-89-3 |
DC7132 |
GF 109203X
Featured
GF109203X is a potent PKC inhibitor with IC50 of 20 nM, 17 nM, 16 nM, and 20 nM for PKCα, PKCβI, PKCβII, and PKCγ, respectively, showing more than 3000-fold selectivity for PKC as compared to EGFR, PDGFR and insulin receptor. |
133052-90-1 |
DC21043 |
GGTI 2417
Featured
GGTI 2417 is the methyl ester prodrug of GGTI-2418, a highly potent, competitive, and selective inhibitor of GGTase I. |
501010-05-5 |
DC21044 |
GGTI 2418
Featured
GGTI 2418 (PTX 100) is a highly potent, competitive, and selective peptidomimetic inhibitor of geranylgeranyltransferase I (GGTI) with IC50 of 9.5 nM, displays 5,600-fold selectivity over FTase. |
501010-06-6 |
DC21042 |
GGTI-2147
Featured
GGTI-2147 is a non-thiol peptidomimetic that inhibits GGTase I and blocks geranyl-geranylation of Rap1A (IC50=0.5 uM). |
191102-87-1 |
DC11246 |
Ghrelin agonist HM01
Featured
Ghrelin agonist HM01 is a novel potent, orally available ghrelin (GHS-R) agonist with Ki of 1.42 nM (human GHS-R1a), induces potent activation of intracellular calcium signaling with EC50 of 1.25 nM. |
1394860-28-6 |
DC10883 |
GI254023X
Featured
GI254023X is a potent MMP9 and ADAM10 inhibitor with IC50s of 2.5 and 5.3 nM, respectively. |
260264-93-5 |
DC10490 |
GIBH-130
Featured
GIBH-130 is a novel inhibitor of neuroinflammation effective in Alzheimer’s disease models. |
1252608-59-5 |
DC7432 |
Givinostat (ITF2357)
Featured
Givinostat (ITF2357) is a potent HDAC inhibitor for maize HD2, HD1B and HD1A with IC50 of 10 nM, 7.5 nM and 16 nM. Phase 1/2. |
732302-99-7 |
DC10081 |
GJ103
Featured
GJ103 is an active analog of the read-through compound GJ072. |
1459687-89-8 |
DC10080 |
GJ103 (sodium salt)
Featured
GJ103 sodium salt is an active analog of the read-through compound GJ072. |
1459687-96-7 |
DC9855 |
GK921
Featured
GK921 is a transglutaminase 2 (TGase 2) inhibitor with average GI50 of 0.9 uM in cancer cell lines. |
1025015-40-0 |
DC8118 |
GKT137831(Setanaxib)
Featured
GKT137831 is a novel and specific dual Nox1/Nox4 inhibitor with Ki of 140±40 nM and 110±30 nM; a potent inhibitor of fibrosis and hepatocyte apoptosis. |
1218942-37-0 |
DC21049 |
Glabrescione B
Featured
Glabrescione B (GlaB) is a small molecule binding to Gli1 zinc finger and impairing Gli1 activity by interfering with Gli1/DNA interaction, inhibits Hh signaling by impairing Gli1 function; inhibits the growth of Hedgehog-dependent tumor cells in vitro and in vivo, inhibits Gli1-dependent growth of cerebellum-derived normal progenitors; inhibits the growth of Gli-dependent medulloblastoma and tumor-derived stem-like cells; inhibits the growth of Gli-dependent basal cell carcinoma in vitro and in vivo. |
65893-94-9 |