GPCR

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Cat. No.	Product Name	Field of Application
DC7781	ML-224 Featured	ML-224 (ANTAG3) is a selective TSH receptor antagonist inhibits stimulation of thyroid function in female mice.
DC10221	MLR-1023	MLR-1023 is a chemical compound which inhibits acid secretion in animal models and also acts as a bronchodilator in histamine-challenged animals.
DC11165	MLS6585	MLS6585 is a novel positive allosteric modulator of the D1 dopamine receptor, potentiatse dopamine-stimulated G-protein- and β-arrestin-mediated signaling and increase the affinity of dopamine for the D1 receptor with low micromolar potencies..
DC3160	Montelukast Sodium Featured	Montelukast belongs to a group of medications known as leukotriene receptor antagonists.
DC10326	Mozavaptan	Mozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM.
DC10437	MRE-269 Featured	MRE-269 is an active metabolite of selexipag, and acts as a selective IP receptor agonist.
DC12258	MRS1186	MRS1186 is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist, with a Ki of 7.66 nM.
DC7203	MRS 2578 Featured	MRS2578 is a potent P2Y6 receptor antagonist with IC50 of 37 nM, exhibits insignificant activity at P2Y1, P2Y2, P2Y4,and P2Y11 receptors.
DC8822	MSX-122 Featured	MSX-122 is a n orally bioavailable inhibitor of CXCR4 with potential antineoplastic and antiviral activities.
DC11270	MSX-130 Featured	MSX-130 is CXCR4 Antagonist.
DC9507	MTEP (hydrochloride)	MTEP Hcl is a potent, selective and non-competitive mGlu5 antagonist with IC50 and Ki of 5 nM and 16 nM, respectively.
DCAPI1550	Naftopidil	Naftopidil is an α-1-Adrenergic receptor antagonist and an antihypertensive.
DC10455	NE-100 Featured	NE100 hydrochloride is a potent and selective σ1 receptor antagonist (Ki = 0.86 nM) that displays > 55-fold selectivity over σ2 receptors and > 6000-fold selectivity over D1,
DCAPI1592	Nebivolol hydrochloride	Nebivolol hydrochloride is a highly selective β1-adrenoceptor antagonist
DC7472	Nedocromil	Nedocromil is an inhaled anti-inflammatory agent for the preventive management of asthma.
DC11469	APD125(Nelotanserin) Featured	Nelotanserin is a potent 5-HT2A inverse agonist, a moderately potent 5-HT2C partial inverse agonist and a weak 5-HT2B inverse agonist, with IC50s of 1.7, 79, 791 nM in IP accumulation assays, respectively.
DC11550	Netazepide	Netazepide (YF476, Sograzepide) is a potent, selective and orally active gastrin/CCK-2 antagonist with IC50 of 0.1 nM.
DC11171	NFEPP	NFEPP is a novel potent, selective pH-dependent μ-opioid receptor (MOR) agonist with a low pKa, shows significantly lower affinity compared with fentanyl at pH 7.4.
DC8836	NIBR189 Featured	NIBR 189 is a potent and selective EBI2 (GPR183) receptor antagonist (IC50 values are 11 and 15 nM for human and mouse EBI2 receptors respectively).
DC10114	Nifenalol Featured	Nifenalol is a beta-adrenoceptor antagonist.
DC9520	NKP608	NKP608 is a non-peptidic derivative of 4-aminopiperidine which acts as a selective, specific and potent antagonist at the neurokinin-1 (NK-1) receptor both in vitro(IC50=2.6 nM) and in vivo.
DC12351	NMI 8739	NMI 8739 is a dopamine D2 autoreceptor agonist, which is an amine conjugate of the DHA carrier and the neurotransmitter dopamine.
DC11386	NNZ-2591 Featured	NNZ2591 (cyclo-L-glycyl-L-2-allylproline)1 is an investigational synthetic analog of cyclic glycine-proline (cGP), a breakdown product of human insulin-like growth factor 1 (IGF-1), that has been chemically modified to increase its half-life, stability, and oral bioavailability.
DC12198	N-Oleoyl glycine	N-Oleoyl glycine is a lipoamino acid, which stimulates adipogenesis associated with activation of CB1 receptor and Akt signaling pathway in 3T3-L1 adipocyte.
DC8583	Asenapine Maleate Featured	Novel psychopharmacologic agent. Displays antagonist activity at 5-HT, dopamine, noradrenalin and histamine receptor subtypes (pKi values are 8.60, 8.40, 10.15, 9.75, 10.46, 8.84, 9.60, 9.94, 8.85, 8.90, 8.84, 9.38, 8.95, 8.93, 8.9, 9.49, 8.91, 9.00 and 8
DC4136	NPS-2143 HCL	NPS 2143 hydrochloride is a selective CaSR (Ca2+-sensing receptor) inhibitor and antagonist, shown to block increases in cytoplasmic Ca2+ concentrations elicited by human Ca2+ receptors expressed in HEK293 cells with an IC50 of 43 nM. NPS 2143 hydrochlori
DC60813	NPS-2143(SB 262470A )	NPS-2143(SB 262470A ) is a selective potent calcium ion-sensing receptor antagonist with IC50 of 43 and 41 nM for cytoplasmic Ca2+ concentrations and parathyroid hormone secretion, respectively.
DC11269	MSX-127（NSC23026） Featured	NSC-23026, also known as MSX-127, is a CXCR4 receptor modulator.
DC7701	NVP-QAV680	NVP-QAV680 is a potent and selective CRTh2 receptor antagonist suitable for clinical testing in allergic diseases.
DC12298	Octreotide acetate (SMS 201-995 (acetate)) Featured	Octreotide acetate, a long-acting synthetic analog of native somatostatin, inhibits growth hormone, glucagon, and insulin more potently.

GPCR

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