| Cat. No. | Product Name | Field of Application | Chemical Structure |
|---|---|---|---|
| DC71780 | Rolapitant hydrochloride | Rolapitant (SCH619734) hydrochloride is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a Ki of 0.66 nM. Rolapitant hydrochloride does not interact with CYP3A4. Rolapitant hydrochloride shows potent anti-emetic activity in a ferret emesis model. |
|
| DC72341 | Septide | Septide ((Pyr6,Pro9)-Substance P) is a potent NK1 receptor agonist with a Kd value of 0.55 nM. |
|
| DC72342 | MEN 10207 | MEN 10207 is a selective NK-2 tachykinin receptor (Neurokinin Receptor) antagonist. MEN 10207 has pA2 values of 5.2, 7.9 and 4.9 in three monoreceptor in vitro assays for NK-1, NK-2 and NK-3 tachykinin receptors, respectively. |
|
| DC72851 | FR 113680 | FR 113680 is a tripeptide substance P antagonist that interacts selectively with the NK1 neurokinin receptor. |
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