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Cat. No. Product Name Field of Application Chemical Structure
DC22096 FT895 FT895 (FT-895) is a potent and selective inhibitor of HDAC11 with IC50 of 3 nM, displays no significant activity against HDAC1-10 (IC50>5 uM).
DC11029 FTBMT Featured FTBMT is a novel selective GPR52 agonist of GPR52, increases intracellular cAMP levels in CHO cells expressing human, mouse, or rat GPR52, with pEC50 of 7.03, 6.85, and 6.87M, respectively.
DC8421 FTI 277 HCl Featured FTI 277 HCl is the methyl ester of FTI 277, which is a potent and selective farnesyltransferase (FTase) inhibitor with IC50 of 500 pM, about 100-fold selectivity over the closely related GGTase I.
DC12537 FtsZ inhibitor C109 FtsZ inhibitor C109 (Compound 10126109) is a broad spectrum antibacterial compound that inhibits the cell division protein FtsZ, inhibits the FtsZ GTPase activity with IC50 of 8.2 uM.
DC3154 Fingolimod HCl(FTY-720) Featured FTY720 (Fingolimod, Gilenya) is a S1P antagonist with IC50 of 0.033 nM.
DC12362 Fuchsine base monohydrochloride Fuchsine base (monohydrochloride) is a magenta dye, which is certified for use for acid-fast staining with carbol-fuchsin.
DC21027 Fumosorinone Fumosorinone is a novel potent, selective protein tyrosine phosphatase SHP2 inhibitor with IC50 of 6.31 uM.
DC11235 Furamidine dihydrochloride Featured Furamidine dihydrochloride (NSC 305831) tyrosyl-DNA phosphodiesterase (Tdp1), also is a selective protein arginine methyltransferase 1 (PRMT1) inhibitor with IC50 of 9.4 uM.
DC10240 Fusidate Sodium Fusidate Sodium is a sodium salt form of fusidic acid, a bacteriostatic antibiotic derived from the fungus Fusidium coccineum and used as a topical medication to treat skin infections.
DC21792 FV-100 FV-100 (Valnivudine, CF-1743) is a potent, selective, bicyclic nucleoside analogue inhibitor of varicella zoster virus (VZV) with EC50 of subnanomolar range in vitro..
DC21031 FzM1.8 FzM1.8 is a small molecule, allosteric agonist of the Frizzled receptor Fzd4 with pEC50 of 6.4, potentiates β-catenin pathway in the absence of any WNT ligand.
DC21032 G 0507 G 0507 is a novel inhibitor of the bacterial LolCDE ABC transporter, binds to LolCDE and stimulates its ATPase activity.
DC21034 G 573 G 573 is a potent and selective, allosteric inhibitor of MEK with Ki of 0.3 nM.
DC11449 G0775 G0775 is a Synethetic analogs of arylomycins.
DC24027 STING Agonist-1(G-10) Featured G10 (STING Agonist 1) is a novel human-specific STING agonist.
DC12300 G3-C12 TFA G3-C12 (TFA) is a galectin-3 binding peptide, with high affinity (Kd) of 88 nM, but shows no affinity for other galectin family members or to other lectins.
DC22548 G-5555 G-5555 is a potent and selective PAK1 inhibitor (Ki=3.7 nM).
DC12438 G6PD activator AG1 Featured G6PD activator AG1 (AG1) is a specific, small molecule that increases the activity of the wild-type, Canton mutant (R459L, EC50=3 uM) and several other common G6PD mutants; displays no effect on the dimerization or activity of several other NAD- or NADP+-dependent dimeric or tetrameric enzymes, including 6PGD, GAPDH, ALDH2, and ALDH3A1; attenuates ROS-induced pericardial edema in a G6PD-dependent manner in zebrafish, reduces hemolysis of human erythrocytes
DC11776 G-744 G-744 is a highly potent, selective inhibitor of BTK with biochemical Ki of 1.28 nM.
DC21035 G907 G907 is a potent, selective small-molecule antagonist of ATP-binding cassette (ABC) transporter MsbA with IC50 of 18 nM.
DC21036 E-72 G9a inhibitor E72 (E-72) is a potent inhibitor of histone H3K9 methyltransferases G9a and G9a-like protein (GLP) with Kd of 136 nM and 164 nM, shows selectivity over the related H3K9 methyltransferase Suv39H2.
DC9381 Gabapentin (hydrochloride) Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog.
DC11053 GAK inhibitor 49 Featured GAK inhibitor 49 is a potent, selective, ATP-competitive inhibitor of cyclin G-associated kinase (GAK, cell IC50=56 nM) with favourable NAK family selectivity (AAK1, STK16, BMP2K).
DC12228 Galactose 1-phosphate Galactose 1-phosphate is an intermediate in the galactose metabolism and nucleotide sugars.
DC12305 Galactose 1-phosphate Potassium salt Galactose 1-phosphate Potassium salt is is an intermediate in the galactose metabolism and nucleotide sugars
DC21038 Galvestine-1 Galvestine-1 is a small molecule MGDG (monogalactosyldiacylglycerol) synthase inhibitor with IC50 of 10 uM by competing with diacylglycerol binding.
DC11071 Gambogenic acid Gambogenic acid (GNA) is a polyprenylated xanthone isolated from gamboge, shows potent antitumor activity and can effectively inhibit the survival and proliferation of cancer cells.
DC12090 Gamitrinib TPP Gamitrinib TPP is a GA mitochondrial matrix inhibitor.
DC9640 gamma-secretase modulator 3 gamma-secretase modulator 3 is a gamma-secretase modulator.
DC21197 Ganaplacide Featured Ganaplacide (KAF156, GNF-156) is a novel antimalarial clinical candidate that shows blood schizonticidal activity with IC50 of 6-17.4 nM against P falciparum drug-sensitive and drug-resistant strains.

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