Novel inhibitors

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Cat. No.	Product Name	Field of Application
DC8631	Framycetin sulphate	Framycetin sulphate
DC9887	FRAX1036 Featured	FRAX1036 is a novel ATP-competitive small molecule inhibitor of group I p21-activated Kinases (PAKs).
DC8003	FRAX-486 Featured	FRAX486 is a selective inhibitor of group I PAKs with IC50s of 8.25/39.5, /55.3 nM for PAK1/PAK2/PAK3 respectivelt; less potent for PAK4(IC50=779 nM).
DC9344	Frentizole	Frentizole, an FDA-approved immunosuppressive drug, is a novel inhibitor of the Aβ-ABAD interaction.
DC20208	Frovatriptan Succinate	Frovatriptan Succinate is the succinate salt form of frovatriptan, a synthetic triptan with serotonin (5-HT) receptor agonist activity especially for the 5-HT1B/1D receptors.
DC21026	FSC 231	FSC 231 (FSC231) is the first, cell-permeable small-molecule inhibitor of PICK1 PDZ domain with Kd of 10.1 uM.
DC23388	FT-001	FT-001 is a novel potent, orally acitve inhibitor of BET bromodomain with IC50 of 0.1 uM for BRD4 BD1.
DC11554	FT-671 Featured	FT-671 is a novel potent, specific, non-covalent USP7 inhibitor with Kd of 65 nM (USP7 catalytic domain).
DC22096	FT895	FT895 (FT-895) is a potent and selective inhibitor of HDAC11 with IC50 of 3 nM, displays no significant activity against HDAC1-10 (IC50>5 uM).
DC11029	FTBMT Featured	FTBMT is a novel selective GPR52 agonist of GPR52, increases intracellular cAMP levels in CHO cells expressing human, mouse, or rat GPR52, with pEC50 of 7.03, 6.85, and 6.87M, respectively.
DC8421	FTI 277 HCl Featured	FTI 277 HCl is the methyl ester of FTI 277, which is a potent and selective farnesyltransferase (FTase) inhibitor with IC50 of 500 pM, about 100-fold selectivity over the closely related GGTase I.
DC12537	FtsZ inhibitor C109	FtsZ inhibitor C109 (Compound 10126109) is a broad spectrum antibacterial compound that inhibits the cell division protein FtsZ, inhibits the FtsZ GTPase activity with IC50 of 8.2 uM.
DC3154	Fingolimod HCl（FTY-720） Featured	FTY720 (Fingolimod, Gilenya) is a S1P antagonist with IC50 of 0.033 nM.
DC12362	Fuchsine base monohydrochloride	Fuchsine base (monohydrochloride) is a magenta dye, which is certified for use for acid-fast staining with carbol-fuchsin.
DC21027	Fumosorinone	Fumosorinone is a novel potent, selective protein tyrosine phosphatase SHP2 inhibitor with IC50 of 6.31 uM.
DC11235	Furamidine dihydrochloride Featured	Furamidine dihydrochloride (NSC 305831) tyrosyl-DNA phosphodiesterase (Tdp1), also is a selective protein arginine methyltransferase 1 (PRMT1) inhibitor with IC50 of 9.4 uM.
DC10240	Fusidate Sodium	Fusidate Sodium is a sodium salt form of fusidic acid, a bacteriostatic antibiotic derived from the fungus Fusidium coccineum and used as a topical medication to treat skin infections.
DC21792	FV-100	FV-100 (Valnivudine, CF-1743) is a potent, selective, bicyclic nucleoside analogue inhibitor of varicella zoster virus (VZV) with EC50 of subnanomolar range in vitro..
DC21031	FzM1.8	FzM1.8 is a small molecule, allosteric agonist of the Frizzled receptor Fzd4 with pEC50 of 6.4, potentiates β-catenin pathway in the absence of any WNT ligand.
DC21032	G 0507	G 0507 is a novel inhibitor of the bacterial LolCDE ABC transporter, binds to LolCDE and stimulates its ATPase activity.
DC21034	G 573	G 573 is a potent and selective, allosteric inhibitor of MEK with Ki of 0.3 nM.
DC11449	G0775	G0775 is a Synethetic analogs of arylomycins.
DC24027	STING Agonist-1(G-10) Featured	G10 (STING Agonist 1) is a novel human-specific STING agonist.
DC12300	G3-C12 TFA	G3-C12 (TFA) is a galectin-3 binding peptide, with high affinity (Kd) of 88 nM, but shows no affinity for other galectin family members or to other lectins.
DC22548	G-5555	G-5555 is a potent and selective PAK1 inhibitor (Ki=3.7 nM).
DC12438	G6PD activator AG1 Featured	G6PD activator AG1 (AG1) is a specific, small molecule that increases the activity of the wild-type, Canton mutant (R459L, EC50=3 uM) and several other common G6PD mutants; displays no effect on the dimerization or activity of several other NAD- or NADP+-dependent dimeric or tetrameric enzymes, including 6PGD, GAPDH, ALDH2, and ALDH3A1; attenuates ROS-induced pericardial edema in a G6PD-dependent manner in zebrafish, reduces hemolysis of human erythrocytes
DC11776	G-744	G-744 is a highly potent, selective inhibitor of BTK with biochemical Ki of 1.28 nM.
DC21035	G907	G907 is a potent, selective small-molecule antagonist of ATP-binding cassette (ABC) transporter MsbA with IC50 of 18 nM.
DC21036	E-72	G9a inhibitor E72 (E-72) is a potent inhibitor of histone H3K9 methyltransferases G9a and G9a-like protein (GLP) with Kd of 136 nM and 164 nM, shows selectivity over the related H3K9 methyltransferase Suv39H2.
DC9381	Gabapentin (hydrochloride)	Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog.

Novel inhibitors

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