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Cat. No. Product name CAS No.
DC22479 Cortisone acetate

Cortisone acetate (Cortisone 21-acetate) is a synthetic glucocorticoid corticosteroid and corticosteroid ester.

50-04-4
DC23908 Cortisone Featured

Cortisone is a pregnane (21-carbon) steroid hormone, one of the main hormones released by the adrenal gland in response to stress.

53-06-5
DC8694 Cortodoxone

Cortodoxone is a glucocorticoid steroid hormone that can be oxygenated to cortisol (Hydrocortisone).

152-58-9
DC9554 Cot inhibitor-1

Cot inhibitor-1 is a COT/Tpl2 inhibitor.

915365-57-0
DC9555 Cot inhibitor-2

Cot inhibitor-2 is a COT/Tpl2 inhibitor.

915363-56-3
DC20933 Cotylimide-VI

Cotylimide-VI (CTL-VI) is a small molecule that perturbs plant hormone strigolactone accumulation and inhibits hypocotyl growth..

419539-64-3
DC10363 Coumestrol Featured

Coumestrol, a phytoestrogen present in soybean products, exhibits activities against cancers, neurological disorders, and autoimmune diseases. It suppresses proliferation of ES2 cells with an IC50 of 50 μM.

479-13-0
DC21413 Cowanin

Cowanin is a novel natural product from Garcinia speciosa that inhibits the Notch signaling pathway with IC50 of 2.4 uM.

21044-85-9
DC8543 CP465022 HCl

CP 465022 hydrochloride is a selective GluR (AMPA) antagonist which is non-competitive.

199655-36-2
DC23320 CP 31398 dihydrochloride Featured

CP-31398 is a small molecule p53 reactivator that protects p53 from thermal denaturation, not only reactivates mutant p53 but also induces stabilization of wild type p53.

1217195-61-3
DC23610 CP-339818 hydrochloride Featured

CP-339818 is a potent, selective, non-peptide KV1.3 channel antagonist with IC50 of 200 nM.

478341-55-8
DC23415 CP-481715

CP-481715 is a potent and selective CCR1 antagonist with Ki of 9.2 nM and IC50 of 74 nM, lacks intrinsic agonist activity and .

212790-31-3
DC4132 CP-547632 Featured

CP-547632 is as a potent inhibitor of the VEGFR-2 and basic fibroblast growth factor (FGF) kinases (IC50 11 and 9 nM, respectively).

252003-65-9
DC8251 CP-724,714

CP-724,714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >640-fold selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc. Phase 2.

383432-38-0
DC8892 CP724714

CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >640-fold selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc in cell-free assays. Phase 2.

537705-08-1
DC9317 CP-809101 (hydrochloride)

CP-809101 Hcl is a potent and selective 5-HT2C receptor agonist with pEC50 of 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors respectively.

1215721-40-6
DC9385 CPA inhibitor

CPA inhibitor is a potent inhibitor for carboxypeptidase A (CPA).

223532-02-3
DC23544 CPG-52364

CPG-52364 (CPG52364) is an orally available, small molecule TLR7/8/9 antagonist for the treatment of systemic lupus erythematosus and other autoimmune disorders..

1093135-60-4
DC7564 CPI 0610(Pelabresib) Featured

CPI 0610 is a potent, selective, and cell-active BET bromodomain inhibitor with IC50 of 39 nM for BRD4-BD1 in TR-FRET assay.

1845726-14-8
DC8002 CPI-360 (R) Featured

CPI-360 is a compound in design and preparation of wew palladium precatalysts for C-C and C-N cross-coupling reactions.

1802175-06-9
DC10527 Ciforadenant (CPI-444) Featured

CPI-444 is an orally administered antagonist of the adenosine A2A receptor. It is designed to block the action of adenosine that is produced by tumors.

1202402-40-1
DC22874 CPI644

CPI644 is a potent, selective, cell-active CBP/EP300 bromodomain inhibitor with IC50 of 0.18 uM for CBP.

1904647-34-2
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