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Other Targets

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Cat. No. Product Name Field of Application Chemical Structure
DC12148 Hosenkoside B Hosenkoside B is a baccharane glycoside isolated from the seeds of impatiens balsamina.
DC12152 Hosenkoside F ((+)-Hosenkoside F) Hosenkoside F is a baccharane glycoside isolated from the seeds of impatiens balsamina.
DC12153 Hosenkoside K Hosenkoside K is a baccharane glycoside isolated from the seeds of impatiens balsamina.
DC12149 Hosenkoside M ((+)-Hosenkoside M) Hosenkoside M is a baccharane glycoside isolated from the seeds of impatiens balsamina.
DC23978 hPGDS-IN-1 Featured hPGDS-IN-1 is a potent, selective hPGDS inhibitor with IC50 of 12 nM in FP or EIA assays..
DC23894 HPI-1 Featured HPI-1 is a Hedgehog (Hh) pathway inhibitor that suppresses signaling through Shh (IC50=1.5 uM) without significantly affecting Wnt signaling (IC50>30 uM).
DC12616 HS-152 HS-152 (HS152) is a specific small-molecule inhibitor of SMAD ubiquitin regulatory factor 1 (SMURF1), not only potently inhibits SMURF1-mediated RHOB degradation with IC50 of 3.2 uM, but also strongly blocks SMURF1-mediated RHOA and SMAD1 degradation (IC5
DC7426 HS-173 Featured HS-173 is a potent PI3Kα inhibitor with IC50 of 0.8 nM.
DC12632 HS220 Featured HS220 (HS-220) is a Plasmodium-selective takinib analog that targets atypical P. falciparum protein kinase 9 (PfPK9, Kd=4.1 uM) but does not inhibit HsTAK1, decreases K63-linked ubiquitination in P. falciparum; inhibits P. berghei parasite load in HuH7 ce
DC21124 HS-38 Featured HS-38 is a potent and selective DAPK1 and DAPK3 (ZIPK) inhibitor with IC50 of 200 nM for DAPK1 and Kd of 280 nM for ZIPK, also inhibits Pim3 (IC50=200 nM), and displays no activity against Src or Abl, little activity against EGFR;
DC23784 HS-72 HS-72 is an allosteric, selective, cell-permeable inhibitor of inducible Hsp70 (Hsp70i or Hsp72), shows selectivity for Hsp70i over the closely related Hsc70 as well as the broader purinome.
DC21126 HSD 1169 HSD1169 is a potent, dual FLT3/TOPK inhibitor with activity against FLT3-ITD secondary mutations (D835 or F691, Kd=1-5 nM), potently inhibits acute myeloid leukemia cell lines (IC50=5 nM).
DC21125 HSD992 HSD992 is a potent, selective CDK2/3 inhibitor with moderate CDK9 inhibition with IC50 of 18 nM, 57 nM and 49 nM for CDK3/cyclin E, CDK2/cyclin A1 and CDK2/cyclin E, respecively.
DC20064 HSK0935 (HSK-0935; HSK 0935) HSK0935 is a potent, highly selective and orally available SGLT2 inhibitor with an IC50 of 1.3 nM. Antihyperglycemic activities.
DC12508 hSMG-1 inhibitor 11e hSMG-1 inhibitor 11e is a potent, selective hSMG-1 kinase inhibitor with IC50 of <0.05 nM, >900-fold selectivity over mTOR, and no significant activity against CDK1/2..
DC12451 hSMG-1 inhibitor 11j hSMG-1 inhibitor 11j is a potent, selective hSMG-1 kinase inhibitor with IC5 0of 0.11 nM, 455-fold selectivity over mTOR and no activity against CDK1/2.
DC20408 HSP27 inhibitor J2 HSP27 inhibitor J2 is a small molecule functional inhibitor of Hsp27, induces significant abnormal HSP27 dimer formation in cancer cells.
DC23794 HSP70 modulator 115-7c HSP70 modulator 115-7c is an artificial co-chaperone, enhancer of Hsp70, stimulats the ATPase and protein-folding activities of a prokaryotic Hsp70 (DnaK) and partially compensated for a Hsp40 loss-of-function mutation in yeast.
DC21149 HT-0712 HT-0712 (IPL-455903) is a novel potent, selective PDE4 inhibitor with IC50 of 0.15 uM for PDE4D3, without effect on PDE1B, PDE3A, and PDE10A.
DC21791 hTG2 inhibitor VA4 hTG2 inhibitor VA4(VA4) is a novel potent, irreversible inhibitor of human tissue transglutaminase (hTG2) with Ki of 12.9 uM, allosterically abolishs its GTP binding ability with a high degree of selectivity and efficiency.
DC20409 HTH-01-091 HTH-01-091 is a potent and selective, cell-permeable, ATP-competitive MELK inhibitor with biochemical IC50 of 10.5 nM.
DC9960 HTHQ Featured HTHQ, which is a hydroquinone monoalkyl ether, is a potent anti-oxidative agent, even at low dose levels.
DC21128 HTS 01037 HTS01037 is a highly potent ligand of adipocyte fatty acid binding protein (A-FABP/aP2) with Ki of 0.67 uM.
DC20081 H-Val-Pro-Pro-OH Featured H-Val-Pro-Pro-OH is a tripeptide derived from milk proteins, specifically a proline-rich peptide, and is known for its inhibitory activity against Angiotensin I Converting Enzyme (ACE). ACE is a key enzyme in the renin-angiotensin system (RAS), which regulates blood pressure by converting angiotensin I to angiotensin II, a potent vasoconstrictor. Inhibition of ACE leads to reduced angiotensin II levels, resulting in vasodilation and lowered blood pressure.
DC10580 hVEGF-IN-1 Featured hVEGF-IN-1 represses human VEGF-A translation and shows antitumor activity.
DC20281 Hycanthone Featured Hycanthone, the most potent mutagen in a series of nine thiaxanthenones, is a potent inducer of nuclear immunoreactivity to antinucleoside antibodies in HeLa cells.
DCAPI1149 Hydralazine HCl Hydralazine HCl
DC20410 Hydrazinocurcumin Featured Hydrazinocurcumin is a synthetic curcumin derivative that inhibits the proliferation of bovine aortic endothelial cells (BAECs) with IC50 of 520 nM without cytotoxicity, inhibits STAT3 phosphorylation and downregulates an array of STAT3 downstream targets.
DCAPI1269 Hydrochlorothiazide Hydrochlorothiazide
DCAPI1198 Hydrocortisone (Cortisol) Hydrocortisone (Cortisol)

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