Cat. No. | Product name | CAS No. |
DC23934 |
FTI-277
Featured
A peptide mimetic of the C-terminal Cys-Val-Ile-Met of K-Ras4B that potently inhibits FTase (Farnesyltransferase) with IC50 of 0.5 nM. |
170006-73-2 |
DC20311 |
Apraglutide
Featured
A peptidic glucagon like peptide 2 (GLP-2) analogue for treatment of type2 diabetes.. |
1295353-98-8 |
DC24173 |
Tolfenpyrad
A pesticide agent.. |
129558-76-5 |
DC22952 |
(S) 93-31
A pH-dependent, GluN2B-selective inhibitor of NMDA receptor with IC50 of 0.19 uM at pH6.9, 10-fold selecivity over brain tissue pH 7.6 (IC50=1.8 uM). |
457897-98-2 |
DC24170 |
TBHQ
A phenolic antioxidant and a selective inducer and activator of Nrf2 that ameliorates doxorubicin-induced cardiotoxicity in vivo. |
1948-33-0 |
DC22501 |
Fosamprenavir calcium
A phosphate ester prodrug of the HIV-1 protease inhibitor amprenavir with improved solubility.. |
226700-81-8 |
DC22845 |
Disoxaril
A picornavirus replication inhibitor by binding to the hydrophobic pocket within the VP1 coat protein, thus stabilizing the virion and blocking its uncoating.. |
87495-31-6 |
DC22620 |
Tiadinil
A plant activator of systemic acquired resistance, boosts the production of herbivore-induced plant volatiles. |
223580-51-6 |
DC5895 |
Apigenin
A plant flavonoid that has been found to inhibit cell proliferation by arresting the cell cycle at the G2/M phase. |
520-36-5 |
DC5880 |
Piceatannol
A plant metabolite possessing anti-leukemic activity; inhibits the non-receptor kinases, Syk and Lck. |
10083-24-6 |
DC22782 |
MDL-72527
Featured
A polyamine oxidase (PAO) inhibitor that inhibits spermine oxidase and N1-acetylpolyamine oxidase with IC50 of 6.1 and 0.02 uM, respectively. |
93565-01-6 |
DC22387 |
Nystatin
A polyene antifungal antibiotic that works by disrupting the cell membrane of the fungal cells.. |
1400-61-9 |
DC22957 |
RU-TRAAK-1
A poorly reversible TRAAK inhibitor, shows no activity for non-K2P channels (Kv1.2, Slo1 and GIRK2).. |
328034-85-1 |
DC22647 |
NU-7163
A poten and selective, ATP-competitive DNA-PK inhibitor with IC50 of 0.19 uM, Ki of 24 nM. |
503468-03-9 |
DC20911 |
Omuralide
Featured
A potent 20S proteasome inhibitor with IC50 of 49 nM (inhibition of proteasomal chymotrypsin-like proteolytic activity).. |
154226-60-5 |
DC21726 |
TAK-802
A potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM. |
263248-16-4 |
DC21727 |
TAK-802 hydrochloride
A potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM. |
263248-36-8 |
DC11614 |
ENT1-IN-39
A potent adenosine transport activity of ENT-1 with IC50 of 26.9 nM. |
2097508-70-6 |
DC20957 |
TCDD
A potent AHR (aryl hydrocarbon receptor) agonist that induces degradation of AhR by the ubiquitin-proteasome pathway. |
1746-01-6 |
DC23997 |
Aleglitazar
A potent and balanced dual PPARα/γ agonist (EC50= 50/21 nM). |
475479-34-6 |
DC22969 |
BC-54
A potent and biologically-active PDE4/7 inhibitor with IC50 of 50-100 nM for PDE4A/B/D, and 140 nM for both PDE7A/B. |
534579-04-9 |
DC20804 |
BMS-204352
A potent and effective calcium-sensitive opener of maxi-K potassium channels (maxi-K) with EC50 of 392 nM at -48.4 mV in HEK293 isolated outside-out membrane patches. |
187523-35-9 |