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PIP-199

  Cat. No.:  DC40328   Featured
Chemical Structure
622795-76-0
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More than 5000 active chemicals with high quality for research!
Field of application
PIP-199 is a selective inhibitor of RMI (RecQ-mediated genome instability protein) core complex/MM2 interaction, with an IC50 of 36 μM. MM2 is the binding site of RMI complex on Fanconi anemia complementation group M protein (FANCM). PIP-199 can be used for the research of sensitizing resistant tumors to DNA crosslinking chemotherapeutics.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 622795-76-0
Chemical Name: PIP-199
Synonyms: ST50111005;ethyl 4-((1-hydroxy-2-phenyl-1H-indol-3-yl)(pyridin-2-yl)methyl)piperazine-1-carboxylate;ethyl 4-[(1-hydroxy-2-phenylindol-3-yl)-2-pyridylmethyl]piperazinecarboxylate;PIP-199;PIP-199 ethyl 4-((1-hydroxy-2-phenyl-1H-indol-3-yl)(pyridin-2-yl)methyl)piperazine-1-carboxylate
SMILES: ON1C2C=CC=CC=2C(=C1C1C=CC=CC=1)C(C1C=CC=CN=1)N1CCN(C(=O)OCC)CC1
Formula: C27H28N4O3
M.Wt: 456.536226272583
Purity: >98%
Sotrage: Powder-20°C3 years4°C2 yearsIn solvent-80°C6 months -20°C1 month
MSDS
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COA
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