Home > Inhibitors & Agonists > GPCR > Adrenergic Receptor
Cat. No. Product name CAS No.
DCAPI1701 Indacaterol Maleate

Indacaterol is an ultra-long-acting β-adrenoceptor agonist with pKi of 7.36.

753498-25-8
DC8914 Indacaterol

Indacaterol(Onbrez; Arcapta) is an ultra-long-acting β-adrenoceptor agonist.

312753-06-3
DC8996 Isoprenaline HCl

Isoprenaline Hydrochloride is a non-selective beta-adrenergic agonist and structurally similar to adrenaline.

51-30-9
DC8987 L-Methyldopa

L-(-)-α-Methyldopa hydrate is an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive drug used as a sympatholytic or antihypertensive.

41372-08-1
DC8714 Levobetaxolol hydrochloride Featured

Levobetaxolol hydrochloride is a beta-adrenergic receptor inhibitor (beta blocker), used to lower the pressure in the eye in treating conditions such as glaucoma.

116209-55-3
DCAPI1580 Medetomidine

Medetomidine hydrochloride is a potent and highly selective α2-AR adrenoceptor agonist (Ki values are 1.08 and 1750 nM for α2- and α1-adrenoceptors respectively). Shows greater selectivity over α1-adrenoceptors than clonidine and UK 14,304 (1620-, 220- an

86347-14-0
DC9191 Metoprolol tartrate

Metoprolol is a cardioselective β1-adrenergic blocking agent.

56392-17-7
DC3172 Mirabegron Featured

Mirabegron is a selective β3-adrenoceptor agonist with EC50 of 22.4 nM.

223673-61-8
DCAPI1550 Naftopidil

Naftopidil is an α-1-Adrenergic receptor antagonist and an antihypertensive.

57149-07-2
DCAPI1592 Nebivolol hydrochloride

Nebivolol hydrochloride is a highly selective β1-adrenoceptor antagonist

152520-56-4
DC10114 Nifenalol Featured

Nifenalol is a beta-adrenoceptor antagonist.

5704-60-9
DC8583 Asenapine Maleate Featured

Novel psychopharmacologic agent. Displays antagonist activity at 5-HT, dopamine, noradrenalin and histamine receptor subtypes (pKi values are 8.60, 8.40, 10.15, 9.75, 10.46, 8.84, 9.60, 9.94, 8.85, 8.90, 8.84, 9.38, 8.95, 8.93, 8.9, 9.49, 8.91, 9.00 and 8

85650-56-2
DC10384 Olodaterol Featured

Olodaterol (BI1744) is a long acting β2-adrenoceptor agonist with an EC50 of 1.4±0.08 nM.

868049-49-4
DC9248 Olodaterol(BI-1744) hydrochloride Featured

Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors located primarily in the lungs.

869477-96-3
DC9101 Phentolamine mesilate

Phentolamine Mesylate is a nonselective alpha-adrenergic antagonist.

65-28-1
DC10115 Piperoxan hydrochloride Featured

Piperoxan hydrochloride is an α2 adrenoceptor antagonist.

135-87-5
DC11138 Guanabenz acetate

R15A inhibitor.

23256-50-0
DC12250 RS 17053 hydrochloride (RS-17053)

RS 17053 hydrochloride is a potent and selective α1A adrenoceptor antagonist, with a pKi value of 9.1 in native cell membrane and a pA2 value of 9.8 in functional assays.

169505-93-5
DC11346 Salbutamol (hydrochloride) Featured

Salbutamol is an agonist of the β2-adrenergic receptor (β2-AR; Kd = 759 nM in a radioligand binding assay using CHO cells expressing the human receptor).

50293-90-8
DC8436 Salmeterol Xinafoate Featured

Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptoms.

94749-08-3
DC8610 Salmeterol Featured

Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptoms.

89365-50-4
DCAPI1485 Silodosin Featured

Silodosin(Rapaflo) is an α1-adrenoceptor antagonist with high uroselectivity. Silodosin causes practically no orthostatic hypotension (in contrast to other α1 blockers). Since Silodosin is a highly selective inhibitor of the α1A adrenergic receptor, it ca

160970-54-7
Page 2 / Total 7 FirstPrevNextLastGoto