| Cat. No. | Product Name | Field of Application | Chemical Structure |
|---|---|---|---|
| DC10386 | Tenapanor Featured | Tenapanor is an inhibitor of the Na+/H+ exchanger NHE3 with IC50 values of 5 and 10 nM against human and Rat NHE3, respectively. |
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| DC9609 | Terutroban Featured | Terutroban is a thromboxane/prostaglandin endoperoxide receptor antagonist. |
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| DC1101 | Ticagrelor (Brilinta,AZD6140) Featured | Ticagrelor is the first reversibly binding oral P2Y12 receptor antagonist, also inhibits CYP2C9 and 4-hydroxylation with IC50 of 10.5 μM and 8.2 μM respectively. |
|
| DC9489 | Tirofiban (hydrochloride monohydrate) Featured | Tirofiban hydrochloride monohydrate is a potent non-peptide, glycoprotein IIb/IIIa (integrins alphaIIbbetaIII) antagonist |
|
| DC7327 | Tirofiban(L700462;MK383) Featured | Tirofiban(L700462;MK383) is a potent non-peptide, glycoprotein IIb/IIIa (integrins alphaIIbbetaIII) antagonist. |
|
| DC7519 | Torcetrapib Featured | Torcetrapib is a CETP inhibitor with IC50 of 37 nM, elevates HDL-C and reduces nonHDL-C in plasma. Phase 3. |
|
| DCAPI1452 | Valsartan | Valsartan is a nonpeptide angiotensin II AT1-receptor antagonist with an IC50 ranging from 39.5 to 116 μM. This in turn causes blood vessel dilation. |
|
| DC8916 | Vanoxerine dihydrochloride Featured | Vanoxerine 2 Hcl(GBR12909) is a potent and selective DRI (Dopamine reuptake inhibitor). |
|
| DC7699 | VTP-27999 Featured | VTP-27999 is an alkyl amine Renin inhibitor; VTP-27999 is useful for Hypertension and End-Organ Diseases. |
|
| DC7040 | WAY-362450 (XL335; Turofexorate isopropyl) Featured | WAY-362450 (XL335; Turofexorate isopropyl) is a highly potent, selective, and orally active farnesoid X receptor (FXR) agonist with an EC50 of 4 nM.WAY-362450 is useful for dyslipidemia. |
|
| DC7753 | Zatebradine hydrochloride | Zatebradine hydrochloride is a bradycardic agent that creates use-dependent inhibition of hyperpolarization-activated current (If) in sinoatrial node cells (EC50 = 480 nM) and Purkinje fibres. |
|
| DC9461 | Zatebradine | Zatebradine(UL-FS49) is a potent HCN channels antagonist, which decreased the heartbeat in a reversible manner; 92% inhibition of the hHCN1-mediated current at 10 uM. |
|
| DC9113 | Ketanserin |
|
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| DC9178 | Ketanserin Tartrate |
|
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| DC8860 | Vorapaxar Featured | Vorapaxar (SCH 530348) is a potent and orally active thrombin receptor (PAR-1) antagonist with Ki of 8.1 nM. |
|
| DC8901 | Azilsartan medoxomil Featured | Azilsartan medoxomil(TAK 491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. |
|
