DCC2874 |
Jxl069 |
Novel potent mitochondrial pyruvate carrier (MPC) inhibitor to treat hair loss |
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DCC2875 |
Jy-1-106 |
Novel BH3 α-helix mimetic, inducing apoptosis in a subset of cancer cells (lung cancer, colon cancer and mesothelioma) by disrupting Bcl-xL and Mcl-1 protein-protein interactions with Bak |
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DCC2876 |
Jyl-1511 |
High-affinity partial agonist of the vanilloid receptor |
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DCC2877 |
Jyl-273 |
Potent TRPV1 agonist |
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DCC2878 |
Jyl-79 |
Potent vanilloid receptor (VR1) agonist |
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DCC2879 |
Jy-xhe-053 |
Selective modulator of GABAA receptors containing the α5 subunit |
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DCC2880 |
Jz-4109 |
Novel β-Glucocerebrosidase modulator, promoting dimerization of β-glucocerebrosidase and revealing an allosteric binding site, stabilizing wild-type and N370S mutant GCase and increases GCase abundance in patient-derived fibroblast cells |
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DCC2881 |
Jz-5029 |
Novel irreversible β-Glucocerebrosidase modulator |
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DCC2882 |
jzad-iv-22 |
Inhibitor of all three monoamine transporters |
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DCC2883 |
Jzp-430 |
Potent, highly selective, and irreversible ABHD6 Inhibitor |
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DCC2884 |
K00135 |
Novel potent and selective inhibitor of PIM kinases |
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DCC2885 |
K00518 |
Novel dual CLK1 and CLK3 inhibitor |
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DCC2886 |
K103 Hydrochloride |
Novel inhibitor of peptidoglycan synthesis targeting the lipid II precursor |
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DCC2887 |
K-14585 |
Novel antagonist for proteinase-activated receptor 2 (PAR2) |
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DCC2888 |
K4610422 |
Novel norditerpenoid inhibitor of testosterone-5α-reductase |
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DCC2889 |
K-8008 |
Novel inhibitor of the interaction of the N-terminally truncated RXR |
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DCC2890 |
K-8012 |
Novel inhibitor of the interaction of the N-terminally truncated RXR |
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DCC2891 |
Kaempulchraol P |
Natural anti-inflammatory agent, inhibiting the NF-κB-mediated transactivation of a luciferase reporter gene, IL-6 production, and COX-2 expression |
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DCC2892 |
Kaempulchraol Q |
Natural anti-inflammatory agent, inhibiting the NF-κB-mediated transactivation of a luciferase reporter gene, IL-6 production, and COX-2 expression |
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DCC2893 |
Kalb001 |
Novel mGlu4 ligand |
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DCC2894 |
Kar425 |
Novel antimalarial agent, providing protection to malaria-infected mice |
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DCC2895 |
Kasugamycin |
Antibiotic, binding within the mRNA channel of the 30S subunit and inhibiting protein synthesis |
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DCC2896 |
Kb130015 |
Novel activator of hERG1 potassium channels, blocking native and recombinant hERG1 channels at high voltages, but activating them at low voltages |
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DCC2897 |
Kbh-a42 |
Novel histone deacetylase inhibitor |
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DCC2898 |
Kbjk557 |
Novel Plk1 PBD inhibitor, showing a remarkable in vitro anticancer effect by inducing Plk1 delocalization, mitotic arrest, and apoptosis in HeLa cells |
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DCC2899 |
Kb-nb165-09 |
Selective inhibitor of Protein_kinase_D1>protein kinase D (PKD); Inhibitor of cell adhesion and HIV; Inhibitor of herpes simplex virus type 1 replication |
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DCC2900 |
Kbp-088 |
Novel highly potent dual amylin and calcitonin receptor agonist (DACRA), showing long-lasting improvement of food preference and body weight loss |
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DCC2901 |
Kb-r7785 |
Novel ADAM12 and MMP inhibitor, ameliorating cardiac function in a transverse aortic constriction (TAC) model by inhibiting the proteolytic activation of HB-EGF signaling, exerting its antidiabetic effect by ameliorating insulin sensitivity through the in |
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DCC2902 |
Kc-11404 |
LTB4 inhibitor for the treatment of b-cell leukemias and lymphomas, potently inhibiting histamine, platelet activating factor,and 5-lipoxygenase |
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DCC2903 |
Kca075 |
Highly specific transglutaminase 2 (TG2) inhibitor |
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