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Cat. No. Product name CAS No.
DC9588 Dofequidar (fumarate)

Dofequidar fumarate(MS-209 fumarate), an orally active quinoline compound, has been reported to overcome MDR by inhibiting ABCB1/P-gp, ABCC1/MDR-associated protein 1, or both.

153653-30-6
DC9323 Dalasetron (Mesylate hydrate)

Dolasetron(MDL-73147) is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy.

878143-33-0
DC3155 Donepezil hydrochloride Featured

Donepezil is a specific and potent AChE inhibitor for bAChE and hAChE with IC50 of 8.12 nM and 11.6 nM , respectively.

120011-70-3
DC11103 Tavapadon Featured

Tavapadon is a potent, orally-bioavailable, selective partial agonist of the dopamine D1 and D5 receptors.

1643489-24-0
DC9308 Doravirine (MK-1439) Featured

Doravirine (MK-1439) is a non-nucleoside reverse transcriptase inhibitor.

1338225-97-0
DC20365 Dorrigocin A

Dorrigocin A is a natural compound that shows potent antiproliferative effect on tumor cell line..

158446-29-8
DC4219 Dorzolomide hydrochloride

Dorzolamide HCl is a carbonic anhydrase inhibitor.

130693-82-2
DC20057 Dot1L-IN-1

Dot1L-IN-1 is a highly potent, selective and structurally novel Dot1L inhibitor with a Ki of 2 pM.

2088518-50-5
DC21895 DOTA-ADIBO

DOTA-ADIBO is a Click Chemistry intermidate used for antibody-drug conjugates..

1374865-01-6
DC10313 Dovitinib lactate

Dovitinib(CHIR-258; TKI258) lactate is a potent inhibitor of fibroblast growth factor receptor 3 (FGFR3) with an IC50 of 5 nM.

692737-80-7
DC9597 Doxapram (hydrochloride hydrate)

Doxapram hydrochloride hydrate inhibits TASK-1, TASK-3, TASK-1/TASK-3 heterodimeric channel function with EC50 of 410 nM, 37 μM, 9 μM, respectively.

7081-53-0
DC23775 DPA-714

DPA-714 is a potent, selective ligand for the translocator protein (TSPO) with Ki of 7.0 nM.

958233-07-3
DC11173 DRAinh-A250 Featured

DRAinh-A250 is a specific inhibitor of Cl-/anion exchanger SLC26A3 (DRA), fully and reversibly inhibits SLC26A3-mediated Cl- exchange with HCO3-, I-, and thiocyanate (SCN-) with IC50 of ~0.2 uM.

858747-13-4
DC20366 DRAK2-IN-16

DRAK2-IN-116 is a potent, selective DRAK2 inhibitor with IC50 of 3 nM, shows weak inhibition for DRAK1 (IC50=51 nM) and no significant activity against DAPK1/2/3 (IC50>1 uM)..

871837-60-4
DC20103 D-Ribose(mixture of isomers) Featured

D-Ribose(mixture of isomers) is an energy enhancer, and acts as a sugar moiety of ATP, and widely used as a metabolic therapy supplement for chronic fatigue syndrome or cardiac energy metabolism. D-Ribose(mixture of isomers) is active in protein glycation

50-69-1
DC20967 DRI-C21045

DRI-C21045 is a novel small-molecule inhibitor of CD40-CD40L protein-protein interaction with IC50 of 0.17 uM in cell-based assays.

2101765-81-3
DC10919 DRP1 inhibitor 4

DRP1 inhibitor 4 is a selective, small molecule inhibitor of the mammalian mitochondrial division dynamin, DRP1 with IC50 of 1.0 uM, shows no activity against OPA1 and DYN1 (IC50>100 uM)..

DC12598 DRV1 (GPR32) agonist C2A

DRV1 (GPR32) agonist C2A (NCGC00135472) is a synthetic molecule that activate human resolvin D1 receptor DRV1/GPR32 receptor with EC50 of 0.37 uM and 0.05 uM in β-arrestin and cAMP assays, respectively.

862811-76-5
DC20968 DS-1040

DS-1040 (DS1040) is a small molecule inhibitor of the activated thrombin-activatable fibrinolysis inhibitor (TAFIa) with IC50 of 1.7 ng/mL for rabbit TAFIa.

1335138-62-9
DC20969 DS-1040 tosylate

DS-1040 tosylate (DS1040) is a small molecule inhibitor of the activated thrombin-activatable fibrinolysis inhibitor (TAFIa) with IC50 of 1.7 ng/mL for rabbit TAFIa.

1335138-89-0
DC20970 DS-1040 tosylate hydrate

DS-1040 tosylate hydrate (DS1040) is a small molecule inhibitor of the activated thrombin-activatable fibrinolysis inhibitor (TAFIa) with IC50 of 1.7 ng/mL for rabbit TAFIa.

1335138-90-3
DC20974 DS16570511

DS16570511 is a cell-permeable inhibitor of the mitochondrial calcium uniporter (MCU) that inhibits serum-induced mitochondrial Ca2+ influx in HEK293A cells with IC50 of 7 uM.

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