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Cat. No.	Product Name	Field of Application
DC33343	SKF-81297 HBr	SKF-81297 HBr is a selective dopamine D1 receptor agonist, which stimulates motor behaviour of MPTP-lesioned monkeys.
DC33344	SKF-83959 HBr	SKF-83959 HBr is a dopamine D1-like receptor partial agonist (Ki values are 1.18, 7.56, 920 and 399 nM for rat D1, D5, D2 and D3 receptors respectively). SKF-83959 HBr may act as an antagonist in vivo, producing anti-Parkinsonian effects and antagonizing the behavioral effects of cocaine.
DC33346	SM19712	SM19712 is a nonpeptide endothelin converting enzyme inhibitor.
DC33347	SM 21	SM 21 is a novel sigma(2) antagonist.
DC33348	SNAP5089	SNAP5089 is a subtype-selective α1A-adrenoceptor antagonist that displays > 600-fold selectivity over other adrenoceptors (Kivalues are 0.35, 220, 370, 540, 800 and 1200 nM for α1A, α1B, α2C, α1D, α2B and α2A subtypes respectively and 540 nM for L-type Ca2+ channels).
DC33349	SQ-29548	SQ-29548 is a highly selective TP receptor antagonist which binds to the human recombinant TP receptor with a Ki of 4.1 nM. SQ-29548 inhibits the aggregation of washed human platelets induced by U-46619 with an IC50 of 0.06 μM.
DC33351	SSR 146977	SSR 146977 is a new potent nonpeptide tachykinin NK3 receptor antagonist.
DC33352	TG6-129	TG6-129 is an antagonist of the EP2 receptor, suppressing PGE2-induced elevation of cAMP in cells expressing EP2 with an IC50 value of 1.6 μM. It is without effect on EP4, DP1, IP, and β2-adrenergic receptors. TG6-129 reduces the expression of COX-2, IL-1β, IL-12, IL-23, IL-6, and TNF-α induced by the EP2-selective agonist butaprost in P388D1 macrophages.
DC33353	U69593	U69593 is a a selective KOR-1 (κ1-opioid receptor) agonist. U-69593 is known to inhibit cocaine sensitization in meso-limbic dopamine neurons by normalizing basal overflow of dopamine.
DC33354	VRT-532	VRT-532 is a CFTR modulator for the treatment of cystic fibrosis.
DC33355	VU0285683	VU0285683 is a negative allosteric modulator of mGlu5 receptors. VU0285683 acts as a full antagonist and blocks the glutamate response to mGlu5 (IC50 = 24.4 nM). VU0285683 is selective for mGlu5 over mGlu1, mGlu3 and mGlu4.
DC33356	DCPIB	DCPIB is a novel Inhibitor of Volume-Regulated Anion Channels, Distinctly Modulating K2P Channels.
DC33357	VU0424465	VU0424465 is a potent mGlu5 positive allosteric modulator and agonist
DC33358	WB 4101	WB 4101 hydrochloride is a α1A-adrenergic selective antagonist.
DC33359	WIN 64338 hydrochloride	WIN 64338 hydrochloride is a potent, non-peptide, competitive bradykinin B2 receptor antagonist.WIN 64338 inhibits [3H]-bradykinin binding on guinea pig trachea with nanomolar affinity but is not active in the rabbit aorta (the classical bradykinin B1 preparation).
DC33360	XAP044	XAP044 is a potent and selective mGlu7 antagonist (IC50 = 88 nM). It inhibits lateral amygdala long term potentiation (LTP) in brain slices from wild type mice. XAP044 displays no effects on the LTP of mGlu7 deficient mice.
DC33361	YM976	YM976 is an orally active PDE4 inhibitor (IC50 = 2.2 nM). YM976 has low emetogenic activity, suggested to be due to poor brain penetration.
DC33362	YS121	YS121 is a dual inhibitor of microsomal prostaglandin E2 synthase-1 and 5-lipoxygenase.
DC33363	ZK93423	ZK93423 is a potent benzodiazepine receptor agonist (IC50 = 1 nM). ZK93423 is non-selective between α1-, α2-, α3- and α5-subunit containing GABAA receptors (Ki values are 4.1, 4.2, 6 and 4.5 nM for inhibition of [3H]Ro15-1788 binding to human recombinant α1β3γ2, α2β3γ2, α3β3γ2 and α5β3γ2 receptors respectively).
DC33364	ZK93426	ZK93426 is a potent, selective and competitive benzodiazepine receptor antagonist (IC50 values are 0.4 and 0.7 nM for inhibition of [3H]-flunitrazepam binding to rat cerebellum and hippocampus respectively)
DC33365	C620-0696	C620-0696 is a novel potent inhibitor of bromodomain PHD-finger transcription factor (BPTF).
DC33366	COH34 S-dioxide	COH34 S-dioxide is an oxidized analog of COH34
DC33367	CRBN-6-5-5-VHL	CRBN-6-5-5-VHL is a novel cell-permeable, potent and selective cereblon degrader.
DC33368	NPE-caged-HPTS	NPE-caged-HPTS is a caged fluorescent pH indicator, rapidly releasing the fluorophore HPTS (pKa 7.25) upon two-photon excitation (>3000 s-1).
DC33369	MRK-740	MRK-740 is a novel potent (IC50: 80?±?16?nM), selective and cell-active PRDM9 inhibitor, specifically and directly inhibiting H3K4 methylation at endogenous PRDM9 target loci.
DC33370	Niclosamide-olamine	Niclosamide-olamine is a Insect Attractant, Repellent and Chemosterilant.
DC33371	Nafcillin sodium	Nafcillin sodium is an antibacterial chemical.
DC33372	Oxacillin sodium	Oxacillin (trade name Bactocill) is a narrow-spectrum beta-lactam antibiotic of the penicillin class developed by Beecham. It was patented in 1960 and approved for medical use in 1962. Oxacillin is a penicillinase-resistant β-lactam. It is similar to methicillin, and has replaced methicillin in clinical use.
DC33373	Levothyroxine sodium	Levothyroxine sodium is a thyroid hormone.
DC33374	Garcinoic Acid	Garcinoic Acid is a natural and selective agonist of pregnane X receptor.

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