| DC34613 |
Ac Phe-NH2 |
Ac-Phe-NH2 is a non-competitive inhibitor (Ki = 8 ± 1.2 mM) of polyubiquitin chain elongation by destabilizing the active trimer. |
|
| DC34614 |
TI 435 |
Clothianidin is an insecticide which acts as an agonist of acetylcholine, thereby stimulating nAChR and activating post-synaptic acetylcholine receptors but not inhibiting AChE. |
|
| DC34615 |
Epiberberine Chloride |
Epiberberine Chloride is a natural anticancer agent which stabilizes telomeric G4s and inhibits telomerase, specifically recognizing the hybrid-2 telomeric G4 predominant in physiologically relevant K+ solution and converts other telomeric G4 forms to hybrid-2. |
|
| DC34616 |
NADA-green |
NADA-green is a fluorescent D-amino acid for labeling peptidoglycans in live bacteria. |
|
| DC34617 |
ONO-8711 |
ONO-8711 is a selective EP1 antagonist. |
|
| DC34618 |
Galloflavin Potassium |
Galloflavin Potassium is an inhibitor of lactate dehydrogenase. |
|
| DC34619 |
DTCBPy |
DTCBPy is an efficient thermally activated delayed fluorescence (TADF) molecule. |
|
| DC34620 |
DCAI hydrochloride |
DCAI hydrochloride is an inhibitor of nucleotide exchange and nucleotide release, by binding to the pocket adjacent to the Ras-SOS interface. |
|
| DC34621 |
Sulindac Sulfide |
Sulindac Sulfide is a metabolite of sulindac. |
|
| DC34622 |
Gentamicin X2 Sulfate |
Gentamicin X2 Sulfate is a potent premature stop codon readthrough molecule and the common precursor of the gentamicin C antibiotic complex. |
|
| DC34623 |
DBHDA |
DBHDA is a reagent to convert a Cys into a Dha moiety by reacting with a C-terminal Cys residue and thus allowing the use of recombinant Ubl G76C mutants to prepare probes. |
|
| DC34624 |
Bortezomib-pinanediol |
Bortezomib-pinanediol is a prodrug of Bortezomib, as well as a proteasome inhibitor. |
|
| DC34625 |
4-Octyl Itaconate |
4-Octyl Itaconate is a cell permeable activator of Nrf2 which inhibits LPS-induced increases in IL-1β mRNA, HIF-1α, and IL-10 in macrophages. |
|
| DC34626 |
Arzanol |
Arzanol is a positive modulator of brain glycogen phosphorylase. |
|
| DC34627 |
BV 02 |
BV02 is an inhibitor of SFN. It also targets YWHAZ of the 14-3-3 protein family. |
|
| DC34628 |
Salicyl-AMS |
Salicyl-AMS is a MbtA Inhibitors and Antimycobacterial Agent. salicyl-AMS [5'-O-(N-salicylsulfamoyl)adenosine] inhibits M. tuberculosis growth in vitro under iron-limited conditions. |
|
| DC34629 |
Flumethasone 21-acetate |
Flumethasone 21-acetate is an anti-inflammatory corticosteroid. |
|
| DC34630 |
Diflorasone Diacetate |
Diflorasone Diacetate is a topical glucocorticoid with anti-inflammatory and immunosuppressive properties. |
|
| DC34631 |
Isoflupredone Acetate |
Isoflupredone Acetate is a topical anti-inflammatory corticosteroid. |
|
| DC34632 |
MDL800
Featured
|
MDL-800 is a first-in-class cellularly active SIRT6 allosteric activator. |
|
| DC34634 |
VUF6002 |
JNJ-10191584 maleate is a highly selective histamine H4 receptor silent antagonist. |
|
| DC34635 |
INH14
Featured
|
INH14 is a cell permeable inhibitor of IKKα/IKKβ, with IC50s of 8.97 and 3.59 μM, respectively. INH14 inhibits the IKKα/β-dependent TLR inflammatory response. INH14 also inhibits downstream of TAK1/TAB1 and NF-kB pathways. Anti-inflammatory and anti-cancer activity. |
|
| DC34636 |
3 Cl-DPA |
3-Cl-DPA is an activator of cardiac troponin by a mechanism distinct from bepridil or TFP. |
|
| DC34637 |
Rifamycin |
Rifamycin is a natural antibiotic which inhibits prokaryotic DNA-dependent RNA synthesis and protein synthesis, thereby blocking RNA-polymerase transcription initiation. |
|
| DC34638 |
Carboxycinnamic acid bishydroxamide |
CBHA is a histone deacetylase (HDAC) inhibitor which potently induces transformed cell growth arrest and terminal differentiation. |
|
| DC34639 |
Disperse Orange 1 |
DO1, also known as Disperse Orange 1, is an anti-amyloid agent which potently delays both seeded and non-seeded Aβ42 polymerization at substoichiometric concentrations, thereby disrupting preformed fibrillar assemblies of synthetic Aβ42 peptides. |
|
| DC34640 |
6PNG |
6-PNG is a Cav3.2 (T-type) calcium channel blocker. |
|
| DC34641 |
PRX |
Pirenoxine, also known as Catalin, is an anti-cataractogenesis agent which interacts with selenite or calcium ions that have been proven as factors leading to the formation of lens cataract. |
|
| DC34642 |
Valerenic acid |
Valerenic acid is a ?-subunit-dependent GABAA receptor modulator. |
|
| DC34643 |
NSC-175151 |
Cytochalasin E is a natural autophagy inhibitor which enhances chemotherapy-induced cell death. Cytochalasin E is an epoxide-containing analog of Cytochalasin B which potently and selectively inhibits the growth of endothelial cells, thereby impairing angiogenesis and tumor growth. Unlike Cytochalasin A and Cytochalasin B, it does not inhibit glucose transport. |
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