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Cat. No. Product Name Field of Application Chemical Structure
DC20628 ABT-102 ABT-102 is a potent, highly selective, orally active TRPV1 antagonist that inhibits agonist-evoked increases in intracellular Ca(2+) levels with IC50 of 5-7 nM.
DC20629 ABT-107 ABT-107 is a potent and selective α7 nAChR agonist with Ki of 0.2-0.6 nM for rat or human cortex α7 nAChRs.
DC23537 ABT-288 ABT-288 is a potent, selective and competitive antagonist of H3 receptor with Ki of 1.9/8.2 nM for human/rat H3 respectively.
DC7352 ABT-333 Featured ABT-333 is an NS5B non-nucleoside polymerase inhibitor.
DC10049 Tebanicline(ABT-594) Featured ABT-594 represents a novel class of broad-spectrum analgesics whose primary mechanism of action is activation of the neuronal nicotinic acetylcholine receptors.
DC10723 ABT-702 Featured ABT-702 is a potent non-nucleoside adenosine kinase inhibitor (IC50 = 1.7 nM), selective over other sites of adenosine interaction (A1, A2A and A3 receptors, adenosine transporter and adenosine deaminase).
DC9262 ABT-719 Featured ABT-719 is a potent bacterial DNA gyrase inhibitor.
DC9261 ABT-719 HCl Featured ABT-719 is a potent bacterial DNA gyrase inhibitor.
DC20630 ABTL0812 ABTL0812 is a novel first-in-class, small molecule that inhibits the Akt/mTORC1 axis and shows antiproliferative effect on tumor cells.
DC23182 ABX464 Featured ABX464 (ABX-464, ABX 464) is a novel class of anti-HIV small molecule targeting Rev-mediated viral RNA biogenesis, shows dose dependent inhibition of HIV-1 replication in stimulated PBMCs with IC50 of 0.1-0.5 uM.
DC7698 AC 55541 Featured AC 55541 is a potent and selective protease-activated receptor 2 (PAR2) agonist (pEC50 = 6.7) that displays no activity at other PAR subtypes or at over 30 other receptors involved in nociception and inflammation.
DC12577 AC-263093 Featured AC-263093 (AC263093) is a potent, functionally selective neuropeptide FF receptor type 2 (NPFFR2) agonist with pKi of 6.9.
DC20300 AC-4-130 AC-4-130 is a novel, potent STAT5 SH2 domain inhibitor, binds to and efficiently blocks STAT5 activation and subsequent transcriptional activity, shows high selectivity for STAT5 over STAT1 and STAT3.
DC21863 AC5 inhibitor C90 AC5 inhibitor C90 is a novel potent, selective adenylyl cyclase type 5 (AC5) inhibitor with IC50 of 30 nM, >5-fold selectivity over AC2 and AC6 subtypes.
DC12086 AC-55649 Featured AC-55649 is a potent, highly isoform-selective agonist of human RARβ2 receptor, with a pEC50 of 6.9.
DC7700 AC710 Featured AC710, is a potent Globally Selective Inhibitor of Platelet-Derived Growth Factor Receptor-Family Kinases.
DC12492 N-(p-Amylcinnamoyl) anthranilic Acid (ACA) Featured ACA is a cell permeable inhibitor of PLA2,reported to inhibit α-ketoisocaproic acid and glyceraldehyde-induced insulin secretion, as well as glucose-induced insulin secretion.
DC9917 Acacetin Featured Acacetin is an O-methylated flavone found in Robinia pseudoacacia (black locust), Turnera diffusa (damiana),Betula pendula (silver birch),and in the fern Asplenium normale.
DC22280 Acarbose Featured Acarbose is the first identified α-glucosidase inhibitor.
DC11458 Ac-DEVD-pNA(Caspase-3 Substrate) Featured Ac-DEVD-pNA is a colorimetric substrate for caspase-3 (CPP32) (Km=9.7μM) and related cysteine proteases.
DC11359 Caspase-3 Substrate Ac-DNLD-AMC is a fluorogenic caspase-3 substrate.
DC9986 Acebilustat(ZK322) Featured Acebilustat(ZK322) is a potent and selective leukotriene A4 hydrolase inhibitor.
DC10592 ASL 601(Acecainide) Featured Acecainide, also known as N-acetylprocainamide and ASL 601, is the N-acetylated metabolite of procainamide.
DC9127 Acemetacin Acemetacin is a non-steroidal anti-inflammatory drug and a glycolic acid ester of indometacin that is a cyclooxygenase inhibitor.
DCAPI1009 Acetanilide (Antifebrin) Acetanilide (Antifebrin)
DC8978 Acetazolamide Acetazolamide is a potent carbonic anhydrase (CA) inhibitor; best-studied agent for the amelioration of acute mountain sickness (AMS).
DC20115 Acetoacetic acid sodium salt Acetoacetic acid sodium salt is a metabolite of non-esterified fatty acids, involved in the development of human diabetes. Acetoacetic acid sodium salt induces oxidative stress to inhibit the assembly of very low density lipoprotein in bovine hepatocytes.
DC10248 Acetohydroxamic acid Acetohydroxamic acid is an Urease Inhibitor. In the urine, it acts as an antagonist of the bacterial enzyme urease.
DC20151 Acetosyringone Featured Acetosyringone is a phenolic compound from wounded plant cells, enables virA gene which encodes a membrane-bound kinase to phosphorylate itself and activate the virG gene product, which stimulates the transcription of other vir genes and itself. Acetosyri
DC12151 Acetyl Perisesaccharide C Acetyl Perisesaccharide C is an oligosaccharide, which is isolated from the root barks of Periploca sepium.

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