Home > Inhibitors & Agonists > Membrane Transporter/Ion Channel
Cat. No. Product name CAS No.
DC9451 Flumazenil

Flumazenil(Ro 15-1788) is a benzodiazepine antagonist, non-selective for α1, α2, α3 or α5-containing GABAA receptors.

78755-81-4
DC9078 Fluoxetine Hydrochloride Featured

Fluoxetine HCl is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class.

56296-78-7
DC4239 Flupirtine maleate

Flupirtine maleateis a non-opioid, centrally acting analgesia, muscle relaxation and neuroprotection. Currently under a clinical trial (recruiting phase) as a treatment for Multiple Sclerosis and has been used as an analgesic.

75507-68-5
DC10158 Fluralaner Featured

Fluralaner (INN) is a systemic insecticide and acaricide Fluralaner through potent blockage of GABA and L-glutamate gated chloride channels.

864731-61-3
DC6917 Vonoprazan Featured

For the detailed information of Vonoprazan, the solubility of Vonoprazan in water, the solubility of Vonoprazan in DMSO, the solubility of Vonoprazan in PBS buffer, the animal experiment (test) of Vonoprazan, the cell expriment (test) of Vonoprazan, the in vivo, in vitro and clinical trial test of Vonoprazan, the EC50, IC50,and affinity,of Vonoprazan, For the detailed information of Vonoprazan, the solubility of Vonoprazan in water, the solubility of Vonoprazan in DMSO, the solubility of Vonoprazan in PBS buffer, the animal experiment (test) of Vonoprazan, the cell expriment (test) of Vonoprazan, the in vivo, in vitro and clinical trial test of Vonoprazan, the EC50, IC50,and affinity,of Vonoprazan, Please contact DC Chemicals..

881681-00-1
DC10947 FPL64176 Featured

FPL64176 is a potent L-type Ca++ channel activator with EC50 of 16 nM.

120934-96-5
DC9381 Gabapentin (hydrochloride)

Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog.

60142-95-2
DC8954 Gabapentin Featured

Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog. It was originally developed to treat epilepsy, and currently is also used to relieve neuropathic pain.

60142-96-3
DC9859 GAL-021 Featured

GAL-021 is a new intravenous BKCa-channel blocker.

1380341-99-0
DC7130 GBR 12935 dihydrochloride Featured

GBR 12935 is a potent and selective inhibitor of dopamine uptake (KD = 5.5 nM in rat striatal membranes).

67469-81-2
DC10721 Gefapixant(AF-219,MK-7264) Featured

Gefapixant(AF-219,MK-7264) is novel P2X3 receptor antagonist.

1015787-98-0
DC10753 GLPG-1837(ABBV-974) Featured

GLPG-1837(ABBV-974) is a novel cystic fibrosis transmembrane conductance regulator CFTR potentiator.

1654725-02-6
DC11678 GLPG-2222

GLPG-2222 (ABBV-2222, Galicaftor) is a novel potent and efficacious CFTR corrector with EC50 of 5 nM.

1918143-53-9
DC11035 GlyT1 inhibitor 46

GlyT1 inhibitor 46 is a novel potent, selective, orally available inhibitor of glycine transporter-1 (GlyT1) with IC50 of 38 and 21 nM for rat and human GlyT1, respectively.

1820934-93-7
DC10874 GlyT2-IN-1(YODA 1) Featured

GlyT2-IN-1(YODA 1) is a glycine transporters GLYT2 inhibitor.

448947-81-7
DC10907 GNE-131 Featured

GNE-131 is a novel NaV1.7 inhibitor with IC50 0.003uM,improving metabolic stability,efficacy in mouse IEM model at C-plasma <2.8uM.

1629063-81-5
DC11090 GR3027 Featured

GR3027 (Golexanolone) is a GABA-A receptor modulating steroid antagonist that selectively antagonizes the enhanced activation of GABAA receptors by neurosteroids such as allopregnanolone and THDOC.

2089238-18-4
DC8006 GS967(GS-458967) Featured

GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa).

1262618-39-2
DC11280 GSK1016790A Featured

GSK1016790A is a novel and potent TRPV4 channel agonist.

942206-85-1
DC10865 GSK2193874 Featured

GSK2193874 is an orally active, potent, and selective TRPV4 antagonist with IC50 of 2 nM and 40 nM for rTRPV4 and hTRPV4.

1336960-13-4
DC9712 Iinerixibat

GSK2330672 is a highly potent, nonabsorbable ASBT(apical sodium-dependent bile acid transporter) inhibitor (hASBT IC50=42 ± 3 nM) .

1345982-69-5
DC8303 GTS 21 2HCl(DMXBA) Featured

GTS 21 dihydrochloride is a partial agonist of α7 nicotinic acetylcholine receptors (nAChRs); also a weak α4β2 and 5-HT3 antagonist at micromolar concentrations.

156223-05-1
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