Novel activator of ethionamide

Novel EthR inhibitor and ethionamide booster

Novel specific bona fide EthR-inhibitor, boosting ETH 4 times in an intravenously infected TB mice model

Novel CBP/p300 Bromodomains inhibitor, binding BRD4 almost identical to SGC-CBP30

Active metabolite of beclomethasone dipropionate

Fatty Ester for Lipid Research

Novel potent and specific inhibitor of dog gastric lipase (DGL)

Inhibitor of monoamine oxidase; Anti-serotonin agent

Inhibitor of angiotensin-converting enzyme (ACE); Prodrug of benazeprilat

Novel potent PI3K inhibitor, suppressing metastasis of non-small cell lung cancer cells by modulating β-catenin/ZEB1 regulatory loop, blocking AKT phosphorylation

Novel inhibitor of HIV-1 Rev function, also acting as a cytostatic agent with substantial antiretroviral activity

Irreversible and nonselective Monoamine_oxidase_inhibitor>monoamine oxidase inhibitor (MAOI)

Antiandrogen, being effective in the treatment of acne, seborrhea, and hirsutism in women

Potent D2/D4 dopamine receptor antagonist, neuroleptic and antipsychotic

anti-HSV agent

Inhibitor of 4-hydroxyphenylpyruvate dioxygenase (HPPD), acting as a herbicide

Anorectic, primarily promoting weight loss through reduced appetite

Useful pharmaceutical building block

Long-acting calcium-blocking agent with significant anti-anginal activity

Novel antibacterial agent against multidrug-resistant Escherichia coli at low concentrations as 0.007 mM, disintegrating membrane, accelerating ROS accumulation, reducing bacterial metabolism, and intercalating into DNA groove

Novel antibacterial agent against multidrug-resistant Escherichia coli at low concentrations as 0.007 mM, disintegrating membrane, accelerating ROS accumulation, reducing bacterial metabolism, and intercalating into DNA groove

Novel inhibitor of plasma kallikrein