Cat. No. | Product name | CAS No. |
DC21026 |
FSC 231
FSC 231 (FSC231) is the first, cell-permeable small-molecule inhibitor of PICK1 PDZ domain with Kd of 10.1 uM. |
1215849-96-9 |
DC23388 |
FT-001
FT-001 is a novel potent, orally acitve inhibitor of BET bromodomain with IC50 of 0.1 uM for BRD4 BD1. |
1778655-51-8 |
DC11554 |
FT-671
Featured
FT-671 is a novel potent, specific, non-covalent USP7 inhibitor with Kd of 65 nM (USP7 catalytic domain). |
1959551-26-8 |
DC22096 |
FT895
FT895 (FT-895) is a potent and selective inhibitor of HDAC11 with IC50 of 3 nM, displays no significant activity against HDAC1-10 (IC50>5 uM). |
2225728-57-2 |
DC11029 |
FTBMT
Featured
FTBMT is a novel selective GPR52 agonist of GPR52, increases intracellular cAMP levels in CHO cells expressing human, mouse, or rat GPR52, with pEC50 of 7.03, 6.85, and 6.87M, respectively. |
1358575-02-6 |
DC8421 |
FTI 277 HCl
Featured
FTI 277 HCl is the methyl ester of FTI 277, which is a potent and selective farnesyltransferase (FTase) inhibitor with IC50 of 500 pM, about 100-fold selectivity over the closely related GGTase I. |
180977-34-8 |
DC12537 |
FtsZ inhibitor C109
FtsZ inhibitor C109 (Compound 10126109) is a broad spectrum antibacterial compound that inhibits the cell division protein FtsZ, inhibits the FtsZ GTPase activity with IC50 of 8.2 uM. |
|
DC3154 |
Fingolimod HCl(FTY-720)
Featured
FTY720 (Fingolimod, Gilenya) is a S1P antagonist with IC50 of 0.033 nM. |
162359-56-0 |
DC12362 |
Fuchsine base monohydrochloride
Fuchsine base (monohydrochloride) is a magenta dye, which is certified for use for acid-fast staining with carbol-fuchsin. |
632-99-5 |
DC21027 |
Fumosorinone
Fumosorinone is a novel potent, selective protein tyrosine phosphatase SHP2 inhibitor with IC50 of 6.31 uM. |
1879030-70-2 |
DC11235 |
Furamidine dihydrochloride
Featured
Furamidine dihydrochloride (NSC 305831) tyrosyl-DNA phosphodiesterase (Tdp1), also is a selective protein arginine methyltransferase 1 (PRMT1) inhibitor with IC50 of 9.4 uM. |
55368-40-6 |
DC10240 |
Fusidate Sodium
Fusidate Sodium is a sodium salt form of fusidic acid, a bacteriostatic antibiotic derived from the fungus Fusidium coccineum and used as a topical medication to treat skin infections. |
751-94-0 |
DC21792 |
FV-100
FV-100 (Valnivudine, CF-1743) is a potent, selective, bicyclic nucleoside analogue inhibitor of varicella zoster virus (VZV) with EC50 of subnanomolar range in vitro.. |
956483-03-7 |
DC21229 |
FX-11
Featured
FX-11 (LDHA inhibitor FX11) is a cell permeable, selective, reversible, NADH competitive inhibitor of lactate dehydrogenase A (LDHA) with Ki of 50 nM (LDHA subunit M), less potent for LDHB or pLDH. |
213971-34-7 |
DC21031 |
FzM1.8
FzM1.8 is a small molecule, allosteric agonist of the Frizzled receptor Fzd4 with pEC50 of 6.4, potentiates β-catenin pathway in the absence of any WNT ligand. |
2204290-85-5 |
DC21032 |
G 0507
G 0507 is a novel inhibitor of the bacterial LolCDE ABC transporter, binds to LolCDE and stimulates its ATPase activity. |
1223998-29-5 |
DC21034 |
G 573
G 573 is a potent and selective, allosteric inhibitor of MEK with Ki of 0.3 nM. |
22868-35-5 |
DC11449 |
G0775
G0775 is a Synethetic analogs of arylomycins. |
2098663-92-2 |
DC24027 |
STING Agonist-1(G-10)
Featured
G10 (STING Agonist 1) is a novel human-specific STING agonist. |
702662-50-8 |
DC12300 |
G3-C12 TFA
G3-C12 (TFA) is a galectin-3 binding peptide, with high affinity (Kd) of 88 nM, but shows no affinity for other galectin family members or to other lectins. |
|
DC22548 |
G-5555
G-5555 is a potent and selective PAK1 inhibitor (Ki=3.7 nM). |
1648863-90-4 |
DC12438 |
G6PD activator AG1
Featured
G6PD activator AG1 (AG1) is a specific, small molecule that increases the activity of the wild-type, Canton mutant (R459L, EC50=3 uM) and several other common G6PD mutants; displays no effect on the dimerization or activity of several other NAD- or NADP+-dependent dimeric or tetrameric enzymes, including 6PGD, GAPDH, ALDH2, and ALDH3A1; attenuates ROS-induced pericardial edema in a G6PD-dependent manner in zebrafish, reduces hemolysis of human erythrocytes |
421581-52-4 |