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Cat. No. Product name CAS No.
DC21026 FSC 231

FSC 231 (FSC231) is the first, cell-permeable small-molecule inhibitor of PICK1 PDZ domain with Kd of 10.1 uM.

1215849-96-9
DC23388 FT-001

FT-001 is a novel potent, orally acitve inhibitor of BET bromodomain with IC50 of 0.1 uM for BRD4 BD1.

1778655-51-8
DC11554 FT-671 Featured

FT-671 is a novel potent, specific, non-covalent USP7 inhibitor with Kd of 65 nM (USP7 catalytic domain).

1959551-26-8
DC22096 FT895

FT895 (FT-895) is a potent and selective inhibitor of HDAC11 with IC50 of 3 nM, displays no significant activity against HDAC1-10 (IC50>5 uM).

2225728-57-2
DC11029 FTBMT Featured

FTBMT is a novel selective GPR52 agonist of GPR52, increases intracellular cAMP levels in CHO cells expressing human, mouse, or rat GPR52, with pEC50 of 7.03, 6.85, and 6.87M, respectively.

1358575-02-6
DC8421 FTI 277 HCl Featured

FTI 277 HCl is the methyl ester of FTI 277, which is a potent and selective farnesyltransferase (FTase) inhibitor with IC50 of 500 pM, about 100-fold selectivity over the closely related GGTase I.

180977-34-8
DC12537 FtsZ inhibitor C109

FtsZ inhibitor C109 (Compound 10126109) is a broad spectrum antibacterial compound that inhibits the cell division protein FtsZ, inhibits the FtsZ GTPase activity with IC50 of 8.2 uM.

DC3154 Fingolimod HCl(FTY-720) Featured

FTY720 (Fingolimod, Gilenya) is a S1P antagonist with IC50 of 0.033 nM.

162359-56-0
DC12362 Fuchsine base monohydrochloride

Fuchsine base (monohydrochloride) is a magenta dye, which is certified for use for acid-fast staining with carbol-fuchsin.

632-99-5
DC21027 Fumosorinone

Fumosorinone is a novel potent, selective protein tyrosine phosphatase SHP2 inhibitor with IC50 of 6.31 uM.

1879030-70-2
DC11235 Furamidine dihydrochloride Featured

Furamidine dihydrochloride (NSC 305831) tyrosyl-DNA phosphodiesterase (Tdp1), also is a selective protein arginine methyltransferase 1 (PRMT1) inhibitor with IC50 of 9.4 uM.

55368-40-6
DC10240 Fusidate Sodium

Fusidate Sodium is a sodium salt form of fusidic acid, a bacteriostatic antibiotic derived from the fungus Fusidium coccineum and used as a topical medication to treat skin infections.

751-94-0
DC21792 FV-100

FV-100 (Valnivudine, CF-1743) is a potent, selective, bicyclic nucleoside analogue inhibitor of varicella zoster virus (VZV) with EC50 of subnanomolar range in vitro..

956483-03-7
DC21229 FX-11 Featured

FX-11 (LDHA inhibitor FX11) is a cell permeable, selective, reversible, NADH competitive inhibitor of lactate dehydrogenase A (LDHA) with Ki of 50 nM (LDHA subunit M), less potent for LDHB or pLDH.

213971-34-7
DC21031 FzM1.8

FzM1.8 is a small molecule, allosteric agonist of the Frizzled receptor Fzd4 with pEC50 of 6.4, potentiates β-catenin pathway in the absence of any WNT ligand.

2204290-85-5
DC21032 G 0507

G 0507 is a novel inhibitor of the bacterial LolCDE ABC transporter, binds to LolCDE and stimulates its ATPase activity.

1223998-29-5
DC21034 G 573

G 573 is a potent and selective, allosteric inhibitor of MEK with Ki of 0.3 nM.

22868-35-5
DC11449 G0775

G0775 is a Synethetic analogs of arylomycins.

2098663-92-2
DC24027 STING Agonist-1(G-10) Featured

G10 (STING Agonist 1) is a novel human-specific STING agonist.

702662-50-8
DC12300 G3-C12 TFA

G3-C12 (TFA) is a galectin-3 binding peptide, with high affinity (Kd) of 88 nM, but shows no affinity for other galectin family members or to other lectins.

DC22548 G-5555

G-5555 is a potent and selective PAK1 inhibitor (Ki=3.7 nM).

1648863-90-4
DC12438 G6PD activator AG1 Featured

G6PD activator AG1 (AG1) is a specific, small molecule that increases the activity of the wild-type, Canton mutant (R459L, EC50=3 uM) and several other common G6PD mutants; displays no effect on the dimerization or activity of several other NAD- or NADP+-dependent dimeric or tetrameric enzymes, including 6PGD, GAPDH, ALDH2, and ALDH3A1; attenuates ROS-induced pericardial edema in a G6PD-dependent manner in zebrafish, reduces hemolysis of human erythrocytes

421581-52-4
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